Target Details
| UniProt AC | Q16832 |
|---|---|
| Gene Symbol | DDR2 |
| Protein Name | Discoidin domain-containing receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 233
- Clinical molecules 21
- Avg pChEMBL 7.22
Associated Diseases (1)
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UEPXBTCUIIGYCY
|
8.0 | Kd | 6 | — | |
VDPIYNSZQSYYGQ
|
8.0 | IC50 | 5 | — | |
RZKBSKVRXHFGJG
|
8.0 | IC50 | 3 | — | |
ODPGGGTTYSGTGO
|
8.0 | Kd | 153 | — | |
WFLPERLYBCBHLO
|
8.0 | IC50 | 2 | — | |
YEPVECGOLOSJGA
|
8.0 | IC50 | 2 | — | |
QAHANVZHNDZWSM
|
7.9 | IC50 | 3 | — | |
VAARYSWULJUGST
|
7.9 | Kd | 119 | Yes | |
YZRLWPBYTMKRQR
|
7.9 | IC50 | 11 | — | |
IUGBGEUCXVKGQK
|
7.9 | IC50 | 13 | — | |
UDRCHZMTVKQTAE
|
7.9 | IC50 | 3 | — | |
KUTDZECNFUUAHC
|
7.8 | IC50 | 3 | — | |
OOEIYCDNOQOFJF
|
7.8 | Kd | 2 | — | |
UGRGTNDQCIYUDE
|
7.8 | IC50 | 3 | — | |
HHZIURLSWUIHRB
|
7.8 | IC50 | 57 | Yes | |
SHTNULLAAVPXRC
|
7.8 | IC50 | 4 | — | |
WGMNFJAFXXXRLZ
|
7.8 | IC50 | 4 | — | |
SAAYRHKJHDIDPH
|
7.7 | IC50 | 3 | — | |
CHYCQBZNTKXHMV
|
7.7 | IC50 | 3 | — | |
CJXZIWDVXAJFBP
|
7.7 | IC50 | 3 | — | |
AIYFNBQHQLKULH
|
7.7 | IC50 | 2 | — | |
XFLAQLCDMJRPFH
|
7.7 | IC50 | 2 | — | |
DAAOYHIERMVREX
|
7.7 | IC50 | 3 | — | |
VDVSFLZBRCBQIQ
|
7.6 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.6 | Kd | 154 | — | |
WJEOLQLKVOPQFV
|
7.6 | Kd | 24 | — | |
UXEXYURPAPXPSR
|
7.5 | IC50 | 2 | — | |
BDDFTQKLPQWOLD
|
7.5 | IC50 | 3 | — | |
MVCOAUNKQVWQHZ
|
7.5 | Kd | 54 | Yes | |
YYIDVDRESUYFKM
|
7.5 | IC50 | 3 | — | |
IFVGNYDOUDEVPK
|
7.5 | IC50 | 3 | — | |
OWEGQACAHYGLOT
|
7.5 | IC50 | 3 | — | |
CZCBVFVSSWZKPW
|
7.4 | IC50 | 3 | — | |
LTQIPTSOJUTHQH
|
7.4 | IC50 | 3 | — | |
UQRCJCNVNUFYDX
|
7.4 | Kd | 27 | — | |
TYGZNGFFKJJPJQ
|
7.4 | IC50 | 3 | — | |
WJTJZDOMFKCYEA
|
7.4 | Kd | 6 | — | |
HKSZLNNOFSGOKW
|
7.4 | Kd | 213 | — | |
XZXHXSATPCNXJR
|
7.4 | Kd | 165 | Yes | |
ARCVIRDCNNOJSS
|
7.4 | Ki | 2 | — | |
AUYHJDXKEGVPNX
|
7.4 | Ki | 2 | — | |
FXEZNFCBNZJTKX
|
7.4 | Ki | 2 | — | |
HDUGVQFEYURLKF
|
7.4 | Ki | 2 | — | |
JEXAMDPQBOIWCJ
|
7.4 | Ki | 2 | — | |
LGJSFFXKADZTNP
|
7.4 | Ki | 2 | — | |
NHHQJBCNYHBUSI
|
7.4 | Kd | 220 | — | |
OWRPCKSLYVXUJS
|
7.4 | Ki | 2 | — | |
PKDCZQAKLPJYFN
|
7.4 | Ki | 2 | — | |
DTAKXSCGKBXZTR
|
7.4 | IC50 | 2 | — | |
KVCQTKNUUQOELD
|
7.4 | IC50 | 6 | — |