Target Details
| UniProt AC | Q16832 |
|---|---|
| Gene Symbol | DDR2 |
| Protein Name | Discoidin domain-containing receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 233
- Clinical molecules 21
- Avg pChEMBL 7.22
Associated Diseases (1)
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YFKFMRKJGPZRSA
|
9.3 | IC50 | 2 | — | |
QXIOZIFTPMAING
|
9.1 | IC50 | 17 | — | |
MPASHPJAIUOWCK
|
8.9 | Kd | 9 | — | |
HKSZLNNOFSGOKW
|
8.8 | IC50 | 408 | — | |
DZUFTTMDQLYMBE
|
8.6 | IC50 | 10 | Yes | |
FQZREJPMQAXXHX
|
8.6 | IC50 | 2 | — | |
JJQCGTDHNYRBRY
|
8.6 | IC50 | 2 | — | |
YXARVHZXTQVAOP
|
8.6 | IC50 | 11 | — | |
RCMOSVXHNJUXAI
|
8.6 | IC50 | 2 | — | |
FNKHCCNFMOPNQT
|
8.5 | IC50 | 2 | — | |
AYQXKPMEHPZRKR
|
8.5 | IC50 | 6 | — | |
GJUVRKOUUBDTIC
|
8.5 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
8.5 | IC50 | 102 | Yes | |
ZEOWTGPWHLSLOG
|
8.5 | IC50 | 2 | — | |
ZPVUIOVIUFJGHO
|
8.5 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
BQRHOTLMFJNXLF
|
8.4 | IC50 | 2 | — | |
BLTXKYZVMMSHDA
|
8.4 | IC50 | 2 | — | |
AQSSMEORRLJZLU
|
8.4 | Kd | 34 | Yes | |
YDNKVGSHYQPIMR
|
8.4 | IC50 | 2 | — | |
GGYCEOGBOJBECJ
|
8.3 | IC50 | 2 | — | |
ISFMOWLMGGXLTK
|
8.3 | IC50 | 2 | — | |
IPXKPFIHNPASKD
|
8.3 | IC50 | 2 | — | |
FHPTWZJZWOYCKG
|
8.3 | IC50 | 5 | — | |
YBEMAJSTGUDUQZ
|
8.3 | IC50 | 3 | — | |
AZOXWOCICFEBCQ
|
8.3 | IC50 | 11 | — | |
PCUPJGFLZXOSJC
|
8.3 | IC50 | 2 | — | |
JCNSIZBVFFVTJE
|
8.2 | IC50 | 3 | — | |
MKXRCUBYHISAAL
|
8.2 | IC50 | 2 | — | |
YHFMRNMPLNTYGD
|
8.2 | IC50 | 2 | — | |
YLTBELFOTTYXRF
|
8.2 | IC50 | 2 | — | |
ITMMHAMHNWGMLK
|
8.2 | IC50 | 2 | — | |
VQQKESJQSNYQOP
|
8.2 | IC50 | 3 | — | |
ASVHVPBHDJQEMH
|
8.2 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
8.2 | Kd | 85 | Yes | |
QCFZDYFUWADUJV
|
8.2 | IC50 | 3 | — | |
GXEGTVQATHKFDH
|
8.2 | IC50 | 10 | Yes | |
KQOYBUCRLZDLBE
|
8.2 | IC50 | 3 | — | |
UPXFBKXBRDBIKU
|
8.2 | IC50 | 3 | — | |
UVMSVIJGLODSFN
|
8.2 | IC50 | 3 | — | |
IZKVIUJIUTXIRH
|
8.1 | IC50 | 2 | — | |
GRFIJHUUQLKEBW
|
8.1 | IC50 | 2 | — | |
NFTNUHHJWIJBRN
|
8.1 | IC50 | 3 | — | |
JHKCROCKUJZVRL
|
8.1 | IC50 | 2 | — | |
WRRRUTZYQAQDCB
|
8.1 | IC50 | 3 | — | |
YXCVYRQZUTUYKZ
|
8.1 | IC50 | 3 | — | |
BYQLDKXFUZAGSM
|
8.1 | IC50 | 2 | — | |
OMCAPVOZCPLRRN
|
8.1 | IC50 | 2 | — | |
RRDDKVJWDOIIFN
|
8.1 | IC50 | 3 | — | |
KVTMDRDZMBVWNC
|
8.0 | IC50 | 6 | — |