Target Details
| UniProt AC | Q16816 |
|---|---|
| Gene Symbol | PHKG1 |
| Protein Name | Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 23
- Clinical molecules 9
- Avg pChEMBL 7.31
KEGG Pathways (3)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
9.4 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
9.2 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
9.2 | Kd | 213 | — | |
NXSJMRCTGYTSTK
|
9.0 | Kd | 200 | — | |
KOZFSFOOLUUIGY
|
8.8 | IC50 | 88 | Yes | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
WINHZLLDWRZWRT
|
8.3 | Kd | 201 | Yes | |
ZHOXAGNPCZTRBN
|
7.9 | Kd | 20 | — | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
JRJKATLTRNXYCE
|
7.1 | IC50 | 4 | — | |
CTNPALGJUAXMMC
|
7.1 | Kd | 151 | — | |
CWJLAVRXVFHDSJ
|
6.9 | IC50 | 13 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
YYLKKYCXAOBSRM
|
6.7 | Kd | 191 | — | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
UBPYILGKFZZVDX
|
6.5 | Kd | 130 | Yes | |
GUBJNPWVIUFSTR
|
6.2 | Kd | 103 | — | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 91 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |