Target Details
| UniProt AC | Q16769 |
|---|---|
| Gene Symbol | QPCT |
| Protein Name | Glutaminyl-peptide cyclotransferase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04389 (Peptidase_M28) |
Summary
- Multi-target molecules 203
- Clinical molecules 0
- Avg pChEMBL 7.61
Active Molecules (203)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FODUYAXDTRJXJS
|
7.0 | IC50 | 2 | — | |
HTNQJWFZNICLJL
|
7.0 | IC50 | 2 | — | |
YPNDSGOSXKLDFG
|
7.0 | IC50 | 2 | — | |
LMESNLGRPUNHNQ
|
6.9 | IC50 | 2 | — | |
GNRHHNMWRYYFEU
|
6.9 | IC50 | 2 | — | |
OCWXTISBGDADNF
|
6.9 | IC50 | 2 | — | |
XJHKAGGRAPVBKR
|
6.8 | IC50 | 2 | — | |
CWKFGLGCGSWELQ
|
6.8 | IC50 | 2 | — | |
MQUFDVSINALCLB
|
6.8 | IC50 | 2 | — | |
QFRNCIQPUMAZHY
|
6.8 | IC50 | 2 | — | |
FFSPXJVZHWCWSI
|
6.7 | IC50 | 2 | — | |
OSLHPTXKIPHFMK
|
6.7 | IC50 | 2 | — | |
OHFOSNNXNKJXOL
|
6.7 | IC50 | 2 | — | |
YZCCUHBHNQCWJM
|
6.7 | Ki | 2 | — | |
GEDBSTPYAKXKIP
|
6.7 | IC50 | 2 | — | |
LSZPAASTOYLCQH
|
6.7 | Ki | 2 | — | |
MLNDVJZTLSHMBU
|
6.6 | Ki | 2 | — | |
NWLLOBVYVNVURL
|
6.6 | IC50 | 2 | — | |
IUAIHDZVYOYFBY
|
6.6 | IC50 | 2 | — | |
ZOUIFXFPCBTXDS
|
6.6 | IC50 | 2 | — | |
FSTYEVLASKHVGG
|
6.5 | IC50 | 2 | — | |
PGOIBMREWDPPGV
|
6.5 | IC50 | 2 | — | |
RTWPGCQKPUAQPX
|
6.5 | Ki | 2 | — | |
WUSACXJBMWPPPL
|
6.5 | IC50 | 2 | — | |
MLNIWJTYHTVNRA
|
6.5 | IC50 | 2 | — | |
BNUXNMGESHTNHZ
|
6.4 | IC50 | 2 | — | |
NOUFXHPCDFRAAM
|
6.4 | IC50 | 2 | — | |
DQUXSQPSPPSFDE
|
6.4 | IC50 | 2 | — | |
IRZRHINGOMTLBA
|
6.4 | IC50 | 2 | — | |
KKKDZZRICRFGSD
|
6.4 | Ki | 6 | — | |
PURGSYUYGRNYOZ
|
6.4 | IC50 | 2 | — | |
VSPYYDBQSOJOEX
|
6.4 | IC50 | 2 | — | |
HAOBIGJCGXSZLT
|
6.4 | IC50 | 2 | — | |
DDDQHTFJWSCMIB
|
6.3 | IC50 | 2 | — | |
FVCIDAPPKZURNK
|
6.3 | IC50 | 2 | — | |
ILRZDJBOXJLREG
|
6.3 | Ki | 2 | — | |
AQJNKGBZCBXQCO
|
6.3 | IC50 | 2 | — | |
BGSQCLIXOIYZLH
|
6.3 | IC50 | 2 | — | |
BUZLMDFOCORSAM
|
6.3 | IC50 | 2 | — | |
GAJVQHYKZUAMGZ
|
6.3 | IC50 | 2 | — | |
IWCVUOUWUKEBPP
|
6.3 | IC50 | 2 | — | |
KZDGWBAHVLSIEW
|
6.3 | IC50 | 2 | — | |
OOIATFCRIVBKDJ
|
6.3 | IC50 | 2 | — | |
PTTPDMCOWQYRLU
|
6.3 | IC50 | 2 | — | |
QRANYZULBJBBLZ
|
6.3 | IC50 | 2 | — | |
UJLGYKMRJHUXQB
|
6.3 | IC50 | 2 | — | |
ULOQIJDKFOANLG
|
6.3 | IC50 | 2 | — | |
VIJTYWPDSYWRJX
|
6.3 | IC50 | 2 | — | |
VNSCXZKICWIPNX
|
6.3 | IC50 | 2 | — | |
WSOHRJMAWOBTQF
|
6.3 | IC50 | 2 | — |