Target Details
| UniProt AC | Q16769 |
|---|---|
| Gene Symbol | QPCT |
| Protein Name | Glutaminyl-peptide cyclotransferase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04389 (Peptidase_M28) |
Summary
- Multi-target molecules 203
- Clinical molecules 0
- Avg pChEMBL 7.61
Active Molecules (203)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NCCZTPAUEYQVBJ
|
7.6 | IC50 | 2 | — | |
PYIKBUMOTKYOMC
|
7.6 | IC50 | 2 | — | |
WASGXHUKGPPEBJ
|
7.6 | IC50 | 2 | — | |
DNDCPICAKRBQLZ
|
7.6 | IC50 | 2 | — | |
VHIGKTNQYRIZBD
|
7.6 | IC50 | 2 | — | |
DVPCBCZIJOTSGR
|
7.6 | IC50 | 2 | — | |
KAPYMMWZUYTENA
|
7.6 | IC50 | 2 | — | |
CGSRGHWGAZPOTQ
|
7.5 | IC50 | 2 | — | |
KIFGZTYWFYAIHI
|
7.5 | IC50 | 2 | — | |
SARHCBLBFIBALH
|
7.5 | IC50 | 2 | — | |
GYHUBSYXHAVYDK
|
7.5 | IC50 | 2 | — | |
QGTMZQZRNWWTQE
|
7.5 | IC50 | 2 | — | |
IQKWGFGJTCUJOF
|
7.5 | IC50 | 2 | — | |
KHRTXNMSFDNHIF
|
7.5 | IC50 | 2 | — | |
NQYKGNCQMRKXDJ
|
7.5 | IC50 | 2 | — | |
CCJCWXPFNUMAEX
|
7.5 | IC50 | 2 | — | |
CPBWBVNNSLFCBC
|
7.5 | IC50 | 2 | — | |
GPQHOIQTHKOAGY
|
7.5 | Ki | 2 | — | |
XLOIDRXYQMEUMU
|
7.5 | IC50 | 2 | — | |
XHIKZWOEFZENIX
|
7.4 | Ki | 2 | — | |
BFBNBJPLBLXPFP
|
7.4 | IC50 | 2 | — | |
LJIAMQXFSCERQG
|
7.4 | IC50 | 2 | — | |
AMQXTNLKQTXNJU
|
7.4 | Ki | 2 | — | |
CMIHONFBJHAJNE
|
7.4 | IC50 | 2 | — | |
YAPJFJYUXSGRHO
|
7.4 | Ki | 2 | — | |
JNKDEHUPDHGMQZ
|
7.3 | IC50 | 2 | — | |
ZONFSXMNDBXNOQ
|
7.3 | IC50 | 2 | — | |
RWBBTILXHXLAKS
|
7.3 | IC50 | 2 | — | |
KEHFVDHJXNSSFH
|
7.3 | IC50 | 2 | — | |
MRAYZXUIMSRTEF
|
7.3 | IC50 | 2 | — | |
OVKWACFPXWSZFC
|
7.3 | Ki | 2 | — | |
PKVUKOYFAIHUHI
|
7.3 | IC50 | 2 | — | |
WZFHFDNWCUWEQM
|
7.3 | IC50 | 2 | — | |
SRLVXCDEMJUVFM
|
7.3 | IC50 | 2 | — | |
YYYPJBARIFRERG
|
7.3 | IC50 | 2 | — | |
MJHMPQRUXGJOQO
|
7.2 | IC50 | 2 | — | |
AFZICJRRIMZCEE
|
7.2 | IC50 | 2 | — | |
HHPQPEGOJOSPRD
|
7.2 | IC50 | 2 | — | |
PHDANEKGGBHYPP
|
7.2 | IC50 | 2 | — | |
FZQXMGLQANXZRP
|
7.2 | Ki | 2 | — | |
MZYLSVFGZFWYEJ
|
7.2 | Ki | 2 | — | |
VLEREHYZFOEMLP
|
7.2 | IC50 | 2 | — | |
APLVIWDXFQTBFL
|
7.1 | IC50 | 2 | — | |
GFEJOPINXGSVOC
|
7.1 | IC50 | 2 | — | |
JZGXOCXYUOBLAU
|
7.1 | IC50 | 2 | — | |
FLWZAMIXHXVKOF
|
7.1 | IC50 | 2 | — | |
LDMSFFQWABTLLU
|
7.1 | IC50 | 2 | — | |
PMLBWSRGSGCWEV
|
7.0 | IC50 | 2 | — | |
QPEFMWKITUBULV
|
7.0 | IC50 | 2 | — | |
NSFVYNHWPXUDCU
|
7.0 | IC50 | 2 | — |