Target Details
| UniProt AC | Q16769 |
|---|---|
| Gene Symbol | QPCT |
| Protein Name | Glutaminyl-peptide cyclotransferase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04389 (Peptidase_M28) |
Summary
- Multi-target molecules 203
- Clinical molecules 0
- Avg pChEMBL 7.61
Active Molecules (203)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTYYZLSQXCEJCR
|
9.0 | IC50 | 2 | — | |
HWJQVJLZIHZEQO
|
9.0 | IC50 | 2 | — | |
IOMCBIJSEZIZBR
|
9.0 | IC50 | 2 | — | |
KRFDXYPODWFBGS
|
9.0 | IC50 | 2 | — | |
MCKHPCBMPQSHRQ
|
9.0 | IC50 | 2 | — | |
NESOMGZBZYWHDD
|
9.0 | IC50 | 2 | — | |
QGLAETHTSCZUGQ
|
9.0 | IC50 | 2 | — | |
QNPKHHPEEDLCEQ
|
9.0 | IC50 | 2 | — | |
QPCXGBQJUONQPC
|
9.0 | IC50 | 2 | — | |
RLJGOUJPSFAQTE
|
9.0 | IC50 | 2 | — | |
VJUSNXPSARZYAY
|
9.0 | IC50 | 2 | — | |
VUMJSLNAEAHKDH
|
9.0 | IC50 | 2 | — | |
YZYTUNZDWQEPIU
|
9.0 | IC50 | 2 | — | |
ZCPILGMRHWXUOV
|
9.0 | IC50 | 2 | — | |
BMQIBWRATXMCAP
|
8.7 | IC50 | 2 | — | |
CTDLZCYAIGFNJP
|
8.7 | IC50 | 2 | — | |
CWCLAUCHKSAOON
|
8.7 | IC50 | 2 | — | |
FOBUIQQYBZZKTE
|
8.7 | IC50 | 2 | — | |
GCCYDFCEXIMIFS
|
8.7 | IC50 | 2 | — | |
HTBGYNXUSLNZMU
|
8.7 | IC50 | 2 | — | |
KUKDVBIGJWCVAL
|
8.7 | IC50 | 2 | — | |
LBILEYIPOVROTM
|
8.7 | IC50 | 2 | — | |
RMUNLQZQODBQGR
|
8.7 | IC50 | 2 | — | |
XOTFSNLHTDBHFH
|
8.7 | IC50 | 2 | — | |
CGPVJQLTXFPNDR
|
8.5 | IC50 | 2 | — | |
DGGQLXDEQQZWDD
|
8.5 | IC50 | 2 | — | |
GVYPSVFYPMCRJI
|
8.5 | IC50 | 2 | — | |
HMLFYWDTHBTPFZ
|
8.5 | IC50 | 2 | — | |
LBTLOWMZKJGWOT
|
8.5 | IC50 | 2 | — | |
LHEZDMQEYGOFFS
|
8.5 | IC50 | 2 | — | |
MNXHIAUMMJXWEU
|
8.5 | IC50 | 2 | — | |
MZCNBZUQFDVOSU
|
8.5 | IC50 | 2 | — | |
NAYJFGGCXSBYLI
|
8.5 | IC50 | 2 | — | |
OAUVDQROYWFPEG
|
8.5 | IC50 | 2 | — | |
PWGUERGOPRKPMW
|
8.5 | IC50 | 2 | — | |
SLFVEFOTJOWYHE
|
8.5 | IC50 | 2 | — | |
UFDUUPBUGCKZRV
|
8.5 | IC50 | 2 | — | |
WONMMZPWEVXUHP
|
8.5 | IC50 | 2 | — | |
YATBHZYAOPKVRX
|
8.5 | IC50 | 2 | — | |
ZXYXXWBJHBAEFK
|
8.5 | IC50 | 2 | — | |
DWKOIVNSZJZOOM
|
8.5 | IC50 | 2 | — | |
LUXVBQYXNBNAIG
|
8.4 | IC50 | 2 | — | |
ITTPKXJQYSTZBT
|
8.4 | IC50 | 2 | — | |
IZCLGPVRGZPKEP
|
8.4 | IC50 | 2 | — | |
SOHOBLQKHUJRBX
|
8.4 | IC50 | 2 | — | |
SVQQWYLZJMSHPS
|
8.4 | IC50 | 2 | — | |
XUGBPKZTAXUEFV
|
8.4 | IC50 | 2 | — | |
MXAZSKBTKUGBLI
|
8.3 | IC50 | 2 | — | |
QZJOWXQTOAXNLK
|
8.3 | IC50 | 2 | — | |
CXVKMAQCKOYECP
|
8.3 | IC50 | 2 | — |