Target Details
| UniProt AC | Q16659 |
|---|---|
| Gene Symbol | MAPK6 |
| Protein Name | Mitogen-activated protein kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 120
- Clinical molecules 3
- Avg pChEMBL 8.61
KEGG Pathways (1)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLXYQKJFFSNBSK
|
7.0 | IC50 | 2 | — | |
MOCDOWIFFPUTEE
|
7.0 | IC50 | 2 | — | |
KJDYRXGMEWBQGR
|
6.9 | IC50 | 2 | — | |
SGVCNDYJJOADQM
|
6.9 | IC50 | 2 | — | |
VAARYSWULJUGST
|
6.8 | Kd | 119 | Yes | |
ROVJHCGYIOSFRW
|
6.8 | IC50 | 2 | — | |
DBXXOIIQTTULBZ
|
6.7 | IC50 | 2 | — | |
YEQPDWJRPJMQQH
|
6.7 | IC50 | 2 | — | |
PDJARQSWGDDFHH
|
6.7 | IC50 | 4 | — | |
FKAMZHMNVQECDN
|
6.7 | IC50 | 2 | — | |
NXWXUDHOUKWAQU
|
6.5 | Kd | 16 | — | |
MMJDVHNODDVMPS
|
6.4 | IC50 | 2 | — | |
KDKUVYLMPJIGKA
|
6.3 | Kd | 91 | Yes | |
OUSFTKFNBAZUKL
|
6.3 | Kd | 58 | Yes | |
ANPSVMXNCCSRFZ
|
6.2 | IC50 | 2 | — | |
XISPMPFADBEOOK
|
6.1 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MEMCTQHLJNUYLA
|
6.0 | IC50 | 2 | — |