Target Details
| UniProt AC | Q16654 |
|---|---|
| Gene Symbol | PDK4 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 381
- Clinical molecules 0
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (381)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ISNBTODJGDBLAZ
|
6.5 | IC50 | 2 | — | |
BVQHFOQYLXZHKL
|
6.5 | IC50 | 2 | — | |
NZKPNEZKGRFGOJ
|
6.5 | IC50 | 2 | — | |
XJVOPOWBIDUKFI
|
6.5 | IC50 | 4 | — | |
ZTSYVKWXYINLJV
|
6.5 | IC50 | 4 | — | |
VCQLZAWRWBAQKG
|
6.5 | IC50 | 2 | — | |
AUJRIOZTXXHUGR
|
6.5 | IC50 | 4 | — | |
BQRFDZQRKCARHX
|
6.5 | IC50 | 4 | — | |
BTVCELJQYVYBMY
|
6.5 | IC50 | 4 | — | |
DXULLUCLDXLAEE
|
6.5 | IC50 | 4 | — | |
KCXGMKDIPWGLSK
|
6.5 | IC50 | 4 | — | |
KURLHYDERFSDAV
|
6.5 | IC50 | 4 | — | |
NULXZQHTQSFRHZ
|
6.5 | IC50 | 4 | — | |
PYWNULWLMYXJIE
|
6.5 | IC50 | 4 | — | |
QWHBUKMSQWNPLU
|
6.5 | IC50 | 4 | — | |
REKSHMUIHDBZEL
|
6.5 | IC50 | 4 | — | |
UHLKSPFADXABBK
|
6.5 | IC50 | 4 | — | |
WQBUEPUJTZXCSW
|
6.5 | IC50 | 4 | — | |
XXFAGYMXMCJALN
|
6.5 | IC50 | 4 | — | |
XZGKZXADQIAIAB
|
6.5 | IC50 | 4 | — | |
ZPNZQVNPYMEKML
|
6.5 | IC50 | 4 | — | |
ZQLXLPNBWGVBKS
|
6.5 | IC50 | 4 | — | |
UDNJJABYGHGSGZ
|
6.5 | IC50 | 2 | — | |
XFKGXBZSDIBBEB
|
6.5 | IC50 | 3 | — | |
LHSKWVQEAJUPOG
|
6.4 | IC50 | 4 | — | |
OVUREOQFPBNHNM
|
6.4 | IC50 | 4 | — | |
YWAFKNHDMNEFPA
|
6.4 | IC50 | 2 | — | |
FLCLKDRMVXBLHR
|
6.4 | IC50 | 4 | — | |
CAAKGPRIVJHBKP
|
6.3 | IC50 | 2 | — | |
BXOOMWSWLIGVOJ
|
6.3 | IC50 | 2 | — | |
DTDZLJHKVNTQGZ
|
6.3 | IC50 | 4 | — | |
RPNZGGQCZUXPBC
|
6.2 | IC50 | 4 | — | |
RRFJREZCKIANGM
|
6.2 | IC50 | 2 | — | |
NLHSXYGKBUOFPL
|
6.2 | IC50 | 4 | — | |
ZBCASIFBVICMSH
|
6.1 | IC50 | 4 | — | |
JAOFIBKJPAHQNQ
|
6.1 | IC50 | 4 | — | |
WRKXOYGLVREKOE
|
6.1 | IC50 | 2 | — | |
QGVSLEINXMWQMT
|
6.0 | IC50 | 4 | — | |
AFRYLLNYYFRUKZ
|
6.0 | IC50 | 4 | — | |
AGIRAUWGTYSFEY
|
6.0 | IC50 | 4 | — | |
AIDMBUXHQJQJMB
|
6.0 | IC50 | 4 | — | |
AVIBHWXBXPFMLQ
|
6.0 | IC50 | 4 | — | |
BOCXGAVHERNIED
|
6.0 | IC50 | 4 | — | |
BOGRKBZCGGVGGS
|
6.0 | IC50 | 4 | — | |
BVSMEZQQQTUAMN
|
6.0 | IC50 | 4 | — | |
CBHNHZXDESJXQZ
|
6.0 | IC50 | 4 | — | |
CKCBDRGQGSQRFN
|
6.0 | IC50 | 4 | — | |
CWAXXGRNESDIFD
|
6.0 | IC50 | 4 | — | |
DFBBARPBDNOHIG
|
6.0 | IC50 | 4 | — | |
DRJCGVYRZOBJOV
|
6.0 | IC50 | 4 | — |