Target Details
UniProt ACQ16654
Gene SymbolPDK4
Protein Name[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF10436 (BCDHK_Adom3) PF02518 (HATPase_c)
Summary
  • Multi-target molecules 381
  • Clinical molecules 0
  • Avg pChEMBL 6.84
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (381)
InChIKey pChEMBL Type Targets Clinical
VPMACFXFRUVPQK 7.0 IC50 4
WBZWNTJAWZVNCI 7.0 IC50 4
WEJYENUPPGWUCM 7.0 IC50 4
WEWLWBDTDINJNR 7.0 IC50 4
WKTAYYWOLXTJGL 7.0 IC50 4
WQJHFNBULHHCAT 7.0 IC50 4
WYUKVGVZYSCCDJ 7.0 IC50 4
XBXCLVBYMZQBFQ 7.0 IC50 4
XFLXHBRVXWEPCZ 7.0 IC50 4
XNWFFSUKXSXYOJ 7.0 IC50 4
XRQPVXUTZFDCGK 7.0 IC50 4
XRQPVXUTZFDCGK 7.0 IC50 4
XVLUOKHYAJARDM 7.0 IC50 4
YDTBZYAJXNXQGG 7.0 IC50 4
YKCSCWCEGAZILJ 7.0 IC50 4
YQIDANKABBOUGC 7.0 IC50 4
YTDJEAZYTGIAJJ 7.0 IC50 4
YZOMOQFRSNGZMJ 7.0 IC50 4
YZOMOQFRSNGZMJ 7.0 IC50 4
ZPMRFYJDPARNBL 7.0 IC50 4
ZUZGRFYAGRDPGJ 7.0 IC50 4
ZVFIHSAIQWKOAE 7.0 IC50 4
ZXOPKIJCZPLJBU 7.0 IC50 4
ZXOPKIJCZPLJBU 7.0 IC50 4
ZYAAUDLDGUEAPN 7.0 IC50 4
ZYLSRWYAGYUONP 7.0 IC50 4
CJKPVNLQNOSPAE 7.0 IC50 4
FSMLYTJJLFECDK 7.0 IC50 4
URBQRLTYIDBJQO 7.0 IC50 4
FSMLYTJJLFECDK 7.0 IC50 4
ZWUKNHQASDKHCT 6.9 IC50 4
LCGNLQSOSJFLKR 6.9 IC50 4
ZWUKNHQASDKHCT 6.9 IC50 4
KOAXITXTHITWLT 6.9 IC50 4
NSEKNXMDWSTZJL 6.9 IC50 4
XNGVNSXRRADPSC 6.9 IC50 4
TWRWVLYTPAORIW 6.8 IC50 4
VPETUWRKODTKNY 6.8 IC50 4
CWHNQKPCYFFKDR 6.8 IC50 4
ZOPYDEDEHVUGTC 6.8 IC50 4
LDFLSIZNFQLCDQ 6.8 IC50 4
FUOYLHLTUNTBFV 6.8 IC50 2
GFICNEUSPWSTPP 6.8 IC50 4
LZCHVMYGVHFFSN 6.7 IC50 6
HVZAUSYZLGXKIP 6.7 IC50 4
QRPZFMFZNJHOTN 6.6 IC50 4
GVZALBNYLGZCKU 6.6 IC50 2
GAFYAXXDUJHTEI 6.6 IC50 4
OIXJNJDUOXZNSC 6.6 IC50 2
BTMDJLDUVYTZBI 6.6 IC50 2
2D structure