Target Details
| UniProt AC | Q16654 |
|---|---|
| Gene Symbol | PDK4 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 381
- Clinical molecules 0
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (381)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLWJFRPCKCAMKV
|
7.0 | IC50 | 4 | — | |
LRFWDRILVLEZJM
|
7.0 | IC50 | 4 | — | |
LRFWDRILVLEZJM
|
7.0 | IC50 | 4 | — | |
LSEQOPAXXJYNDG
|
7.0 | IC50 | 4 | — | |
LSJRQFSUVPSXTH
|
7.0 | IC50 | 4 | — | |
LWPVJGVLNMPBPK
|
7.0 | IC50 | 4 | — | |
LWPVJGVLNMPBPK
|
7.0 | IC50 | 4 | — | |
MJDOETCLTIAWPE
|
7.0 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
7.0 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
7.0 | IC50 | 4 | — | |
MMWXYJPJGRRGIT
|
7.0 | IC50 | 4 | — | |
NDZDDEMSENNYBA
|
7.0 | IC50 | 4 | — | |
NMNWEMCMDINIHC
|
7.0 | IC50 | 4 | — | |
NSMJZJFXYGOOET
|
7.0 | IC50 | 4 | — | |
OAODSMWKFRASCR
|
7.0 | IC50 | 4 | — | |
OCVNXALHQSJRLS
|
7.0 | IC50 | 4 | — | |
OFVWPLPGVMYLFN
|
7.0 | IC50 | 4 | — | |
OJZZFYPZMQVSJV
|
7.0 | IC50 | 4 | — | |
OWFZQPQOHDKLNC
|
7.0 | IC50 | 4 | — | |
OYIVLQTWURCFIL
|
7.0 | IC50 | 4 | — | |
OYIVLQTWURCFIL
|
7.0 | IC50 | 4 | — | |
OZPNMFRXHFNHAE
|
7.0 | IC50 | 4 | — | |
PRCTUAYWNHMKTR
|
7.0 | IC50 | 4 | — | |
PSQMYJVREYGDAB
|
7.0 | IC50 | 4 | — | |
PTHJRVBBACHGOH
|
7.0 | IC50 | 4 | — | |
PUPFOOFVPKXKKS
|
7.0 | IC50 | 4 | — | |
QAAAEMHGCDUTQF
|
7.0 | IC50 | 4 | — | |
QEHFXBQCHXZVPP
|
7.0 | IC50 | 4 | — | |
QOBHBSIALHUBML
|
7.0 | IC50 | 4 | — | |
QOMVKWOSNCOMEE
|
7.0 | IC50 | 4 | — | |
QORZJUPQLUQVLM
|
7.0 | IC50 | 4 | — | |
QQEXAKLRPMBVMU
|
7.0 | IC50 | 4 | — | |
QTUKYQAPKFQRDT
|
7.0 | IC50 | 4 | — | |
QVSHTTDOPIXQHK
|
7.0 | IC50 | 4 | — | |
RDZHNFZDJQDIFX
|
7.0 | IC50 | 2 | — | |
RRPLLQMMPJWFIR
|
7.0 | IC50 | 4 | — | |
RRVGEDSKKYXEEQ
|
7.0 | IC50 | 4 | — | |
RWKAWUMWADJEBW
|
7.0 | IC50 | 4 | — | |
SJEXWLLUJGZGAK
|
7.0 | IC50 | 4 | — | |
SQEBZRWBDVPJDR
|
7.0 | IC50 | 4 | — | |
SWUFKVPRVHWIRW
|
7.0 | IC50 | 4 | — | |
SXBULXXRUIFERC
|
7.0 | IC50 | 4 | — | |
SZCHNEBNXWTYGU
|
7.0 | IC50 | 4 | — | |
SZCHNEBNXWTYGU
|
7.0 | IC50 | 4 | — | |
TZKXWAODTKIRQH
|
7.0 | IC50 | 4 | — | |
UDXRPQUWDSCOTK
|
7.0 | IC50 | 4 | — | |
UMRLOUSNWOYFFM
|
7.0 | IC50 | 4 | — | |
UOLOUISPBSPRGG
|
7.0 | IC50 | 4 | — | |
VIRNQTUQCWCOAV
|
7.0 | IC50 | 4 | — | |
VLTVCXJATKADNO
|
7.0 | IC50 | 4 | — |