Target Details
| UniProt AC | Q16644 |
|---|---|
| Gene Symbol | MAPKAPK3 |
| Protein Name | MAP kinase-activated protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 0
- Avg pChEMBL 6.88
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HVXKQKFEHMGHSL
|
8.7 | Kd | 21 | — | |
ZGBAJMQHJDFTQJ
|
7.6 | Kd | 15 | — | |
MUOKSQABCJCOPU
|
7.6 | Kd | 36 | — | |
MIKAKZKNMYZLDX
|
7.3 | Ki | 42 | — | |
CMWRPDHVGMHLSZ
|
7.3 | IC50 | 22 | — | |
JCFJQIHDZHHMQT
|
6.8 | Ki | 42 | — | |
NKGLJTITEFZKAN
|
6.8 | Ki | 35 | — | |
OWFLADWRSCINST
|
6.7 | IC50 | 30 | — | |
IGXJXMLDIIGDNE
|
6.7 | IC50 | 8 | — | |
OWDRQHVEJIYVOI
|
6.6 | Ki | 47 | — | |
UEIRKXUBXCSHJE
|
6.4 | Ki | 19 | — | |
LKUJDAHYLPICSE
|
6.2 | Ki | 24 | — | |
USHMNZBDAOGLMB
|
6.2 | Ki | 26 | — | |
NNQMSHWOTYMSDC
|
6.2 | IC50 | 3 | — | |
HATNHAMXMKJCEI
|
6.1 | Ki | 9 | — |