Target Details
| UniProt AC | Q16620 |
|---|---|
| Gene Symbol | NTRK2 |
| Protein Name | BDNF/NT-3 growth factors receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13855 (LRR_8) PF16920 (LRRCT_2) PF01462 (LRRNT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 538
- Clinical molecules 31
- Avg pChEMBL 7.51
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (538)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KMRRAHVRJDHPQG
|
6.7 | IC50 | 3 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
VNBRGSXVFBYQNN
|
6.7 | IC50 | 22 | Yes | |
AGYRJOAGMDIFKL
|
6.7 | Ki | 17 | — | |
BIKYDWLMTPRSQL
|
6.7 | Ki | 50 | — | |
BLQYVHBZHAISJM
|
6.7 | Ki | 54 | — | |
DKSNLQYRZJKYOC
|
6.7 | Ki | 51 | — | |
IDTRMLOMEBMZLF
|
6.7 | IC50 | 3 | — | |
JISZKDFLHFISOW
|
6.7 | Ki | 6 | — | |
LJKJYKWDLJUZHA
|
6.7 | Ki | 24 | — | |
NWAUBAGBGOPJLF
|
6.7 | Ki | 51 | Yes | |
QBKUOOQFSVMDPB
|
6.7 | Ki | 31 | — | |
RTYJMUXLFRYRBU
|
6.7 | Ki | 35 | — | |
XLFYOIVELARSKP
|
6.7 | Ki | 33 | — | |
ZNMQXOQGTZNCCL
|
6.7 | IC50 | 3 | — | |
ZXLFIHLBHMLHFJ
|
6.7 | Ki | 31 | — | |
KFOUNCZZUSEIAE
|
6.7 | IC50 | 3 | — | |
QKKIWEILHCXECO
|
6.7 | IC50 | 24 | — | |
YWAOBYAAHVVPGD
|
6.7 | IC50 | 3 | — | |
NPVVAEDMCPEANH
|
6.6 | IC50 | 3 | — | |
WIMIUZAOKNILRU
|
6.6 | IC50 | 3 | — | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
DNFPFLPJDNMARR
|
6.6 | IC50 | 3 | — | |
DWRDCEAGIMHGDA
|
6.6 | IC50 | 3 | — | |
ROWJAVCITQHSST
|
6.6 | IC50 | 3 | — | |
LGHBDVLAHHANMX
|
6.6 | Ki | 53 | — | |
VSVWQTDDGQSGHP
|
6.6 | Ki | 51 | — | |
WQFGNANQTYLQBP
|
6.6 | Ki | 16 | — | |
XRPCAAGDYPEUIE
|
6.6 | IC50 | 3 | — | |
ZFCQSGVBHIEECU
|
6.6 | IC50 | 3 | — | |
NXYJKXDQFIZEFL
|
6.6 | IC50 | 3 | — | |
CKFSGFBIQDUWKV
|
6.6 | IC50 | 5 | — | |
UEBRHNWRYCBULZ
|
6.6 | Ki | 2 | — | |
KNZNJSNITSGMNY
|
6.5 | IC50 | 2 | — | |
BKZUKTAHVHZYFR
|
6.5 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 91 | Yes | |
ATGVCJYHNOSZEV
|
6.5 | Ki | 23 | — | |
AYKPYAOQPANRFS
|
6.5 | IC50 | 3 | — | |
BSFNGHCTZDCQBF
|
6.5 | Ki | 93 | — | |
DANNFAQHLGBAQY
|
6.5 | IC50 | 3 | — | |
DOLVPVSWTLFZMQ
|
6.5 | Ki | 17 | — | |
JJGSOVIZOMZMCS
|
6.5 | Ki | 35 | — | |
KSVGVUZJQAEMMJ
|
6.5 | IC50 | 3 | — | |
QLWUDWMYFSWGHK
|
6.5 | Ki | 22 | — | |
RGNHKJWHFIPHIM
|
6.5 | Ki | 66 | — | |
ZVPDNRVYHLRXLX
|
6.5 | Ki | 35 | Yes | |
FOEHDMQTILPVSW
|
6.5 | IC50 | 3 | — | |
LRBMWVVYMSGWJD
|
6.5 | IC50 | 3 | — | |
XFLAQLCDMJRPFH
|
6.5 | IC50 | 5 | — |