Target Details
| UniProt AC | Q16620 |
|---|---|
| Gene Symbol | NTRK2 |
| Protein Name | BDNF/NT-3 growth factors receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13855 (LRR_8) PF16920 (LRRCT_2) PF01462 (LRRNT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 538
- Clinical molecules 31
- Avg pChEMBL 7.51
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (538)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBYBXLWMSCLSKJ
|
7.0 | IC50 | 3 | — | |
PRWFEEBNDGCREE
|
7.0 | IC50 | 3 | — | |
IIJKGBMUSGQZJO
|
7.0 | IC50 | 3 | — | |
VKBFHTIUXUCYRQ
|
7.0 | Ki | 66 | — | |
YTPXNCADDOOFPA
|
7.0 | Kd | 2 | — | |
JRLOPMVTMMPZMV
|
6.9 | IC50 | 3 | — | |
VLHUMLSNFMCPFI
|
6.9 | IC50 | 3 | — | |
GUBJNPWVIUFSTR
|
6.9 | Kd | 103 | — | |
IXZOFWVKCDIGGX
|
6.9 | IC50 | 3 | — | |
KMYBTZOVMXFXAU
|
6.9 | IC50 | 3 | — | |
JREJWPGPNAQDPQ
|
6.9 | IC50 | 3 | — | |
CJUJLGFTKBBDMG
|
6.9 | Ki | 9 | — | |
FLEAYYMORDPWAJ
|
6.9 | Ki | 90 | — | |
HEUSUIRCBWROMH
|
6.9 | Ki | 64 | — | |
HKZKELVPGXJIMW
|
6.9 | Ki | 41 | — | |
IHVVNQIYQOLNQR
|
6.9 | IC50 | 2 | — | |
JXNMCDLXYWQTIW
|
6.9 | Ki | 13 | — | |
MHCPAORAYMTGCZ
|
6.9 | Ki | 37 | — | |
MVJMMLFMPWITEJ
|
6.9 | Ki | 110 | — | |
NRGYZNJPCGRCLV
|
6.9 | Ki | 52 | — | |
QNUKRWAIZMBVCU
|
6.9 | Ki | 46 | — | |
UJBJWYNPUOLFIZ
|
6.9 | IC50 | 49 | — | |
WFTZMAAMCVPJJT
|
6.9 | Ki | 26 | — | |
AJDJDSOIQFUPTC
|
6.9 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.9 | Kd | 231 | Yes | |
BMBZCEYEGICFNU
|
6.9 | IC50 | 3 | — | |
FQGDIYVVDKJSNC
|
6.9 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
6.8 | Kd | 191 | — | |
RALKOVHFGYUBAB
|
6.8 | IC50 | 5 | — | |
TVDCSSYHPQMVIE
|
6.8 | IC50 | 3 | — | |
JCXYIKRACZYAIU
|
6.8 | IC50 | 3 | — | |
OXQTXNVWTNDAQF
|
6.8 | IC50 | 5 | — | |
RIPARGUDVVDTTD
|
6.8 | IC50 | 3 | — | |
AIQDZMUPVYDVLB
|
6.8 | Ki | 48 | — | |
CQBBMNXXVMOFCA
|
6.8 | Ki | 39 | — | |
GSXRCPJTNIGKSZ
|
6.8 | Ki | 43 | — | |
GWMATETWMAQOFL
|
6.8 | Ki | 36 | — | |
HZPACYSNLOCDLW
|
6.8 | Ki | 48 | — | |
NFKMFNBKEOQNPZ
|
6.8 | Ki | 43 | — | |
NHFDRBXTEDBWCZ
|
6.8 | Ki | 41 | — | |
PYXQMJSGJIJHJT
|
6.8 | Ki | 28 | — | |
XBYVOPRDASFDMY
|
6.8 | Ki | 42 | — | |
ZGDSBEUMPIMXBM
|
6.8 | Ki | 42 | — | |
JLXDGCSIJRNQOU
|
6.8 | IC50 | 3 | — | |
NJAVDBDBSBBDKS
|
6.8 | IC50 | 3 | — | |
MTQFLGAYNKVAPI
|
6.8 | IC50 | 4 | — | |
SEZFNTZQMWJIAI
|
6.8 | Ki | 22 | — | |
RBMCJUWMZVILNQ
|
6.7 | IC50 | 3 | — | |
OTBHAYAYGBSHCF
|
6.7 | Kd | 2 | — | |
FTDWSWREBGYXDZ
|
6.7 | IC50 | 10 | — |