Target Details
| UniProt AC | Q16620 |
|---|---|
| Gene Symbol | NTRK2 |
| Protein Name | BDNF/NT-3 growth factors receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13855 (LRR_8) PF16920 (LRRCT_2) PF01462 (LRRNT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 538
- Clinical molecules 31
- Avg pChEMBL 7.51
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (538)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
APPXQUDJLJXULP
|
8.1 | IC50 | 47 | — | |
HDMQHDILMFAMEX
|
8.1 | IC50 | 3 | — | |
HFDYFIJWKPLZKI
|
8.1 | IC50 | 4 | — | |
KZFPHKZQVCYHEZ
|
8.1 | IC50 | 3 | — | |
QNTSEJJXGJAWBN
|
8.1 | IC50 | 3 | — | |
QTSGFRRREQFWGK
|
8.1 | IC50 | 3 | — | |
ADHIYNKWKQQREL
|
8.1 | IC50 | 3 | — | |
DADASRPKWOGKCU
|
8.1 | IC50 | 9 | — | |
FAYAUAZLLLJJGH
|
8.1 | IC50 | 36 | Yes | |
WLAVZAAODLTUSW
|
8.1 | IC50 | 7 | — | |
AYQXKPMEHPZRKR
|
8.0 | IC50 | 6 | — | |
GLRHZMRFCNDDIZ
|
8.0 | IC50 | 3 | — | |
UAZRNUYGVNUMRW
|
8.0 | IC50 | 3 | — | |
BRTHUECZMVKNMQ
|
8.0 | Ki | 31 | — | |
KKYPRNBBPBRJQX
|
8.0 | Ki | 40 | — | |
NIKNJFKATRPZSL
|
8.0 | Ki | 9 | — | |
RBXYGQNZRVPDNB
|
8.0 | Ki | 34 | — | |
WPHKIQPVPYJNAX
|
8.0 | Ki | 81 | — | |
XIWVEZNCIIVZQH
|
8.0 | IC50 | 3 | — | |
XJSFDMGICAWQFS
|
8.0 | Ki | 60 | — | |
ZYEIOSXTPZLYKG
|
8.0 | IC50 | 3 | — | |
KDFREDAEEQQCFD
|
8.0 | IC50 | 3 | — | |
NNDVLAPMFXYAAS
|
8.0 | IC50 | 3 | — | |
WABINVADIAZJHY
|
8.0 | IC50 | 3 | — | |
ZKDXRFMOHZVXSG
|
8.0 | IC50 | 13 | Yes | |
IQEIAIXWJHRRRI
|
7.9 | IC50 | 3 | — | |
YYDUWLSETXNJJT
|
7.9 | IC50 | 5 | — | |
FFCFHBVSGILIJY
|
7.9 | Ki | 17 | — | |
MCCCQFAOMZMZKE
|
7.9 | Ki | 52 | — | |
PTVPBWWDGZSEAF
|
7.9 | Ki | 63 | — | |
IGJZBYFJOGZJQO
|
7.9 | IC50 | 3 | — | |
LZFGLNXIDZGIEG
|
7.9 | IC50 | 3 | — | |
NPZSESRPQGYDMI
|
7.9 | IC50 | 3 | — | |
OIZJENLXXROKNH
|
7.9 | IC50 | 3 | — | |
QXQMNBCLKYICGU
|
7.9 | IC50 | 3 | — | |
SEIMODXPKPYLDQ
|
7.9 | IC50 | 3 | — | |
YGUHZTGUYHUMMF
|
7.9 | IC50 | 3 | — | |
ZBSQPLKGTYVAIB
|
7.9 | IC50 | 3 | — | |
JFSJERWBWSRHJA
|
7.9 | IC50 | 3 | — | |
GEGAHMIBPFSFDY
|
7.8 | IC50 | 3 | — | |
LIGNPDHIOGZBEA
|
7.8 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
XOMSZJJKZWBVAH
|
7.8 | IC50 | 3 | — | |
AUTGNDRENPBZKA
|
7.8 | IC50 | 3 | — | |
FUJQPFBKDKKXHX
|
7.8 | IC50 | 3 | — | |
JZORFWRZZRNPER
|
7.8 | IC50 | 3 | — | |
PHKCNLPGORPBKO
|
7.8 | IC50 | 3 | — | |
HVJJVFGMNLSTHA
|
7.8 | IC50 | 3 | — | |
AUFWLXVVSPEREI
|
7.8 | IC50 | 3 | — | |
COXSWEZHBTXILY
|
7.8 | IC50 | 3 | — |