Target Details
| UniProt AC | Q16620 |
|---|---|
| Gene Symbol | NTRK2 |
| Protein Name | BDNF/NT-3 growth factors receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13855 (LRR_8) PF16920 (LRRCT_2) PF01462 (LRRNT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 538
- Clinical molecules 31
- Avg pChEMBL 7.51
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (538)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HFNKQEVNSGCOJV
|
6.4 | Kd | 65 | — | |
LAJAAZMLLWPYKV
|
6.4 | IC50 | 2 | — | |
OEPYXKHANLDDLG
|
6.4 | IC50 | 2 | — | |
IGRYEDIMNMEBBU
|
6.4 | IC50 | 9 | — | |
KQZFHDUZMBMCMO
|
6.4 | IC50 | 3 | — | |
CXBBWVXSZINRCS
|
6.4 | Ki | 41 | — | |
FUMCKNCUEAQHCV
|
6.4 | Ki | 103 | — | |
KTEIFNKAUNYNJU
|
6.4 | Ki | 48 | — | |
PROLIXHVRCJEFH
|
6.4 | Ki | 46 | — | |
PUPCRRRSBUYJAD
|
6.4 | Ki | 44 | Yes | |
XKFTZKGMDDZMJI
|
6.4 | Ki | 56 | — | |
CIEAJZWSESCRGI
|
6.4 | IC50 | 2 | — | |
YJYPEGFCCCYDKE
|
6.4 | IC50 | 3 | — | |
GSAMVOHLWIOYLH
|
6.3 | IC50 | 2 | — | |
JTYYECWUMLHCSJ
|
6.3 | IC50 | 8 | — | |
HHZIURLSWUIHRB
|
6.3 | Kd | 57 | Yes | |
VGNCTJVAUAZQDJ
|
6.3 | IC50 | 3 | — | |
CNTCGRJDUJEUDG
|
6.3 | Ki | 37 | — | |
IPTSYCYNQJITNJ
|
6.3 | Ki | 12 | — | |
KQSQZFWRXUXPMI
|
6.3 | Ki | 3 | — | |
NOBMKUVHFRVBES
|
6.3 | Ki | 19 | — | |
RWEHAHIEUDLKGT
|
6.3 | Ki | 33 | — | |
TXHOCWWJSGCZLC
|
6.3 | Ki | 18 | — | |
UGUZOLHBLLTLBA
|
6.3 | Ki | 15 | — | |
WUWDLXZGHZSWQZ
|
6.3 | Ki | 41 | — | |
XFWUTMHVDGPWLH
|
6.3 | Ki | 75 | — | |
ZLVOTRRGLSDLPF
|
6.3 | Ki | 36 | — | |
AIWDHNDUIDAYMO
|
6.2 | IC50 | 4 | — | |
JVLYHJYNLHAPID
|
6.2 | IC50 | 3 | — | |
MVCOAUNKQVWQHZ
|
6.2 | Kd | 54 | Yes | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
CVWXJKQAOSCOAB
|
6.2 | Kd | 35 | — | |
ACNCCUVYXQGPKZ
|
6.2 | Ki | 31 | — | |
CAWSIAKYPLHUPL
|
6.2 | IC50 | 2 | — | |
DLWMVUDMPMKGEE
|
6.2 | Ki | 24 | — | |
HRZOUBQYVUXBNS
|
6.2 | Ki | 38 | — | |
MLDQJTXFUGDVEO
|
6.2 | Ki | 85 | Yes | |
MPVGZUGXCQEXTM
|
6.2 | Ki | 61 | Yes | |
NGHPFFZNDYPKNE
|
6.2 | Ki | 2 | — | |
SDBOIBYRBWPIEL
|
6.2 | Ki | 31 | — | |
UXMNYFJHEBEDJS
|
6.2 | Ki | 19 | Yes | |
ZAARMHXLYCHRAK
|
6.2 | Ki | 20 | — | |
YMPWYIHAVYUJEK
|
6.2 | IC50 | 2 | — | |
ODNQXPDPRYQVRN
|
6.2 | IC50 | 4 | — | |
UVJXOGHWHKUVGT
|
6.2 | IC50 | 4 | — | |
PIQCTGMSNWUMAF
|
6.1 | Kd | 137 | Yes | |
QUOOWHZYYXJNSD
|
6.1 | IC50 | 3 | — | |
UXXQOJXBIDBUAC
|
6.1 | Kd | 21 | Yes | |
SZURKEABSBIIMJ
|
6.1 | IC50 | 5 | — | |
FRLSQVCECUJDAT
|
6.1 | IC50 | 2 | — |