Target Details
| UniProt AC | Q16602 |
|---|---|
| Gene Symbol | CALCRL |
| Protein Name | Calcitonin gene-related peptide type 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 123
- Clinical molecules 0
- Avg pChEMBL 9.11
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (123)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RUEPQTQOKXMCFR
|
7.5 | IC50 | 2 | — | |
ANPOMVNSKAJOBS
|
7.4 | IC50 | 2 | — | |
FJVIXLDHHTWOCN
|
7.4 | IC50 | 2 | — | |
PWPMKDORTALZSG
|
7.4 | IC50 | 2 | — | |
DPKUUAZWPCGLJU
|
7.3 | IC50 | 2 | — | |
RUEPQTQOKXMCFR
|
7.3 | IC50 | 2 | — | |
BWLUJBRNLJVDMS
|
7.2 | IC50 | 2 | — | |
YOTPJQUOGGWKAG
|
7.2 | IC50 | 2 | — | |
SQQZSWBNZZDEAJ
|
7.1 | Ki | 2 | — | |
DTYAISJWGQJWJI
|
7.1 | IC50 | 2 | — | |
VDLYRUOYUCCKKR
|
7.0 | IC50 | 4 | — | |
LJKCPRJTSAUESM
|
6.6 | Ki | 2 | — | |
CVPWNBYUSUFFDB
|
6.6 | IC50 | 2 | — | |
RLKYTIXOYWIXQK
|
6.5 | IC50 | 4 | — | |
JXTWPKPSAOKCLS
|
6.4 | IC50 | 4 | — | |
DSMQHSCNENFKPV
|
6.4 | IC50 | 4 | — | |
FFKJRZZAQCOLKI
|
6.3 | IC50 | 2 | — | |
TUXVCNZWFXHVRY
|
6.3 | Ki | 2 | — | |
JNMYUIOIISURGX
|
6.3 | IC50 | 4 | — | |
PORPTQSGGWNOJX
|
6.3 | IC50 | 2 | — | |
FFKJRZZAQCOLKI
|
6.0 | Ki | 2 | — | |
SSWCBXZFRVUVJD
|
6.0 | IC50 | 2 | — | |
BXOQPDIPQMXQDO
|
6.0 | IC50 | 2 | — |