Target Details
UniProt ACQ16602
Gene SymbolCALCRL
Protein NameCalcitonin gene-related peptide type 1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00002 (7tm_2) PF02793 (HRM)
Summary
  • Multi-target molecules 123
  • Clinical molecules 0
  • Avg pChEMBL 9.11
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (123)
InChIKey pChEMBL Type Targets Clinical
RZFPBHZKAKASKU 9.8 Ki 2
VFDRHALOJDLYPX 9.8 Ki 2
XWGGMGIJGQPTMR 9.8 Ki 2
BEUICGVSHZDHTP 9.7 Ki 2
GZNXOZBMUGJEGL 9.7 Ki 2
YYSNPBLETNIGCW 9.7 IC50 2
MKGOTRHHJCVLEJ 9.7 Ki 2
BURSVINJULGQMN 9.7 Ki 2
MNNURILBCATYRI 9.7 Ki 2
NFKNHAHXAMZIFN 9.7 Ki 2
IDKKNSOZWQOAAS 9.6 Ki 4
FUGYGCWFKVNINL 9.6 Ki 2
SKPSTNHVXHTZKY 9.6 Ki 2
YYIRLNHPNVBRKV 9.6 Ki 2
HTLWMOKBJQKDIJ 9.5 IC50 2
DYUUVBPOUOMLAV 9.5 Ki 2
FSDQUSHNPJAZQP 9.5 Ki 2
RYURPNQKLUHMSX 9.4 Kd 2
VSXKCMDTFNFBTN 9.3 Ki 2
UQAIKQPLSLVDNM 9.2 Ki 2
OQNIKHVOMULLTM 9.2 Ki 2
RKADCONIJFEQAL 9.1 Ki 2
OXLJPUYTPSHXLV 9.1 Ki 2
FMRWVSPLSDNMNK 9.1 Ki 2
BMINCMUOYCLAEZ 9.0 Ki 2
WRBNREYWMONIFZ 8.9 Ki 2
TZNQLVLILPGVRT 8.9 IC50 2
YYUSPECBRKLNEH 8.9 Ki 2
WAZDMGGJAWEMTD 8.8 Ki 2
LZESRBNZLWMEIJ 8.7 Ki 2
CRXOAPVFOGTLOS 8.7 Ki 2
SLMBMWIBJWYEMS 8.7 Ki 2
CGDZXLJGHVKVIE 8.7 IC50 3
UXDXGHBXIOBTBN 8.7 Ki 2
CCCSWRIKNOQGJG 8.7 IC50 2
NDACAFBDTQIYCQ 8.6 IC50 4
QEHHKXFWVQCUTL 8.6 Ki 2
CLPPWVGSNJNGGK 8.6 IC50 2
NJLGJIVVVAPJOY 8.5 Ki 2
IDZRBQDLAOIEQP 8.4 Ki 2
TYOGCTPXYBIGHG 8.3 IC50 2
JQBAIBGWHDJVCY 8.3 IC50 2
FMTJCQSCGILGKH 8.1 Ki 2
BZPVIHOWUYCVHT 8.1 Ki 2
CDWIFANGBNPXSD 8.1 Ki 2
WMTZDAHGKCEIAT 8.1 Ki 2
LVJLXLXVWDOXCC 7.9 IC50 4
COFTYEBEOOYCDC 7.8 Ki 2
UGVTUQAEJUZTMQ 7.8 Ki 2
GKEYVYYYUKUCAC 7.5 IC50 2
2D structure