Target Details
UniProt ACQ16602
Gene SymbolCALCRL
Protein NameCalcitonin gene-related peptide type 1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00002 (7tm_2) PF02793 (HRM)
Summary
  • Multi-target molecules 123
  • Clinical molecules 0
  • Avg pChEMBL 9.11
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (123)
InChIKey pChEMBL Type Targets Clinical
WZSCJOMKGFGYAC 11.3 Ki 2
OCUJZNSQSAMOBQ 11.0 IC50 2
MGPZDZUWVWCXMD 11.0 Ki 2
RHWMJBIOLRHWNI 11.0 Ki 2
RFEWOLIROHKSKX 10.8 Ki 2
QIVUCLWGARAQIO 10.8 Ki 2
OPTPGWMNIOROHR 10.8 Ki 2
OVTQOOXOGJZWCA 10.8 Ki 2
GONXFONBYFBWQQ 10.7 Ki 2
ITIXDWVDFFXNEG 10.7 Ki 3
LHCOLCAUMRHKNE 10.7 Ki 2
RFOPIEIJLKLOPX 10.7 Ki 2
AZAANWYREOQRFB 10.7 Ki 3
PDCKQHZWVCORCM 10.6 Ki 2
UJUBRNFNBYNWEZ 10.6 Ki 2
GFOFSWUKCXORBM 10.6 Ki 2
LIPVCPUZWNTQHV 10.5 Ki 2
GWAJYOYPXYSDHT 10.4 Ki 2
HENCBPGDMCRTPM 10.4 Ki 2
JEFZERUDBVOEHW 10.4 Ki 2
LGRBIIARKNGKBN 10.4 Ki 2
VJFRMTZBLLJSOE 10.4 Ki 2
KHYFGYPWDCLESN 10.3 IC50 2
IENHCDUZUNPICI 10.3 Ki 2
XJYAUYAJBKPGJN 10.3 Ki 2
SUKIQFSJOWYYTQ 10.3 Ki 2
LIQMLKRGQPLTKF 10.2 Ki 2
WDLPYUGNINUHRV 10.2 Ki 2
FJQKIFRGRSGWHP 10.2 Ki 2
DDOOFTLHJSMHLN 10.2 Ki 2
HAXMEUJKWQSGEX 10.2 Ki 2
MBRFNJSXLBOYAO 10.1 Ki 2
OJPMDWJBEALLDT 10.1 Ki 2
PIYNZUIYDJFKLR 10.1 Ki 2
WGSUOJIEVHEZAD 10.1 Ki 2
KADHZTQMULOACF 10.1 Ki 2
GQEUXVCWAIGMFG 10.0 Ki 2
GPRUCWKXSWAMFN 10.0 Ki 2
KIHBNAPZVSKRKC 10.0 Ki 2
OIPRTBOJXKHIGX 10.0 Ki 2
QENXEFFSRSLOGM 10.0 Ki 2
UTGSAOCPUHBZKU 10.0 Ki 2
KCXRARVKXIZHRH 10.0 Ki 2
BPUHNEMQLUNYIN 9.9 Ki 2
CUZDSMAQNGFFFO 9.9 Ki 2
GAPKJXGSZQANSF 9.9 Ki 2
GUILBDPDYMIGBQ 9.8 Kd 3
ICNUFHZEIOFOEN 9.8 IC50 2
XLAANMGBSWWGLO 9.8 Ki 2
LREUBQQMJXJGNU 9.8 Ki 2
2D structure