Target Details
| UniProt AC | Q16584 |
|---|---|
| Gene Symbol | MAP3K11 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF14604 (SH3_9) |
Summary
- Multi-target molecules 79
- Clinical molecules 17
- Avg pChEMBL 7.06
KEGG Pathways (2)
Active Molecules (79)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
XLSYZSRXVVCHLS
|
6.6 | Kd | 48 | — | |
DOZKSGRZZQMRCD
|
6.6 | IC50 | 2 | — | |
ZZSBPGIGIUFJRA
|
6.6 | Kd | 46 | — | |
PKGQDPNUCJTZSZ
|
6.6 | IC50 | 2 | — | |
HVVKFYHINSILFO
|
6.5 | IC50 | 11 | Yes | |
PBCZSGKMGDDXIJ
|
6.5 | Kd | 68 | Yes | |
CJQGLUJHMXCLQY
|
6.5 | IC50 | 11 | — | |
CXQHYVUVSFXTMY
|
6.5 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.5 | Kd | 149 | — | |
DCYHJVFMNYSPNT
|
6.5 | IC50 | 9 | — | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
MZDKLVOWGIOKTN
|
6.3 | Kd | 80 | — | |
HCBIATVCCJRSKR
|
6.3 | IC50 | 5 | — | |
OBJNFLYHUXWUPF
|
6.3 | IC50 | 17 | — | |
RWJSBHSWVMKBER
|
6.3 | IC50 | 2 | — | |
VAARYSWULJUGST
|
6.3 | Kd | 119 | Yes | |
YBVSJBLXFZBKSU
|
6.3 | IC50 | 3 | — | |
RHFIAUKMKYHHFA
|
6.2 | IC50 | 9 | — | |
XCOSAQGGGZDYJN
|
6.2 | IC50 | 11 | — | |
GCIKSSRWRFVXBI
|
6.2 | Kd | 109 | Yes | |
XZXHXSATPCNXJR
|
6.2 | Kd | 165 | Yes | |
CUIHSIWYWATEQL
|
6.1 | Kd | 61 | Yes | |
CMJCXYNUCSMDBY
|
6.1 | Kd | 15 | — | |
FWLMVFUGMHIOAA
|
6.0 | Kd | 26 | — | |
BFSMGDJOXZAERB
|
6.0 | Kd | 33 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |