Target Details
| UniProt AC | Q16584 |
|---|---|
| Gene Symbol | MAP3K11 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF14604 (SH3_9) |
Summary
- Multi-target molecules 79
- Clinical molecules 17
- Avg pChEMBL 7.06
KEGG Pathways (2)
Active Molecules (79)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NXSJMRCTGYTSTK
|
8.5 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
8.4 | Kd | 170 | — | |
DFBYFJSXUCUKLA
|
8.2 | IC50 | 2 | — | |
OCMCHCVNRKLMAQ
|
8.2 | IC50 | 4 | — | |
KOZFSFOOLUUIGY
|
8.1 | IC50 | 88 | Yes | |
CVXZWDPKRAIHOI
|
8.0 | IC50 | 4 | — | |
MDAFGVXLBFQEJH
|
8.0 | IC50 | 4 | — | |
NHHQJBCNYHBUSI
|
8.0 | Kd | 220 | — | |
SIBOQVCECFIQAO
|
8.0 | IC50 | 2 | — | |
NHDDTLMPCVOXFH
|
7.9 | IC50 | 16 | Yes | |
KOZFSFOOLUUIGY
|
7.9 | IC50 | 26 | — | |
QKKIWEILHCXECO
|
7.8 | IC50 | 24 | — | |
BMGQWWVMWDBQGC
|
7.8 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.8 | Kd | 91 | Yes | |
UIARLYUEJFELEN
|
7.7 | Kd | 289 | Yes | |
YVKIJUOXNIWLHR
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 49 | Yes | |
GOTKZROZHBWZJH
|
7.7 | IC50 | 6 | — | |
UFLRHQRKTYVKGB
|
7.7 | IC50 | 4 | — | |
RAOJISQDGOOXTK
|
7.7 | IC50 | 14 | Yes | |
SCMLRESZJCKCTC
|
7.6 | IC50 | 7 | — | |
VZJUKEQMHBEIKH
|
7.6 | IC50 | 2 | — | |
WENCWJUIDFEPSK
|
7.6 | IC50 | 3 | — | |
SIHPNVHZKXZMMW
|
7.5 | IC50 | 3 | — | |
NBGYLHIDCLVBHE
|
7.4 | IC50 | 6 | Yes | |
UQHKXSZPEUNUDH
|
7.4 | IC50 | 2 | — | |
LYFDGRJCBMWOKJ
|
7.4 | IC50 | 3 | — | |
MEXUTNIFSHFQRG
|
7.3 | IC50 | 21 | Yes | |
RYYNGWLOYLRZLK
|
7.3 | Kd | 45 | — | |
ASMLDRAEBPYENO
|
7.3 | IC50 | 10 | — | |
DKZYXHCYPUVGAF
|
7.3 | Kd | 112 | — | |
QMLALHXGVBGFIC
|
7.3 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
7.2 | Kd | 97 | Yes | |
XIKCRRWSJXYZMA
|
7.2 | IC50 | 2 | — | |
JJQPROAZGIYDBL
|
7.2 | IC50 | 4 | — | |
HSWWFIPPMAFLPH
|
7.2 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
7.1 | Kd | 50 | — | |
ABMSAGZBJYEZGT
|
7.1 | IC50 | 4 | — | |
SRZPGKHRQCVEAS
|
7.1 | IC50 | 2 | — | |
FPXKTABMRKRDJN
|
7.0 | IC50 | 2 | — | |
GSHILQCUENBVBZ
|
7.0 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
6.9 | IC50 | 92 | — | |
PXLLDBDHYSZSQP
|
6.9 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.9 | Kd | 599 | — | |
CMAAJKFJPMUHEN
|
6.8 | IC50 | 3 | — | |
VFBGXTUGODTSPK
|
6.8 | IC50 | 2 | — | |
BFKOYMDZLSTZJN
|
6.8 | IC50 | 2 | — | |
IJICOKICFQCHBP
|
6.8 | IC50 | 2 | — |