Target Details
| UniProt AC | Q16566 |
|---|---|
| Gene Symbol | CAMK4 |
| Protein Name | Calcium/calmodulin-dependent protein kinase type IV |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 14
- Clinical molecules 5
- Avg pChEMBL 6.48
KEGG Pathways (13)
- Alcoholism
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Apelin signaling pathway
- Calcium signaling pathway
- Cholinergic synapse
- Glioma
- Long-term potentiation
- Longevity regulating pathway
- Neurotrophin signaling pathway
- Osteoclast differentiation
- Oxytocin signaling pathway
- cAMP signaling pathway
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
7.5 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
7.4 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
HFNKQEVNSGCOJV
|
6.7 | Kd | 65 | — | |
MCUJKPPARUPFJM
|
6.4 | Kd | 11 | — | |
KGPGFQWBCSZGEL
|
6.4 | Kd | 59 | Yes | |
AYCPARAPKDAOEN
|
6.4 | Kd | 73 | — | |
HZTYDQRUAWIZRE
|
6.3 | Kd | 40 | Yes | |
VERWOWGGCGHDQE
|
6.2 | Kd | 23 | — | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |