Target Details
| UniProt AC | Q16549 |
|---|---|
| Gene Symbol | PCSK7 |
| Protein Name | Proprotein convertase subtilisin/kexin type 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01483 (P_proprotein) PF00082 (Peptidase_S8) PF16470 (S8_pro-domain) |
Summary
- Multi-target molecules 14
- Clinical molecules 0
- Avg pChEMBL 7.11
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHBJTTGFHCHQHS
|
9.9 | Ki | 6 | — | |
UFNWIBYSOUCSGW
|
7.9 | Ki | 4 | — | |
QDGGHGYNQCXHOK
|
7.8 | Ki | 4 | — | |
PRKRCMZHFKTMTR
|
7.1 | Ki | 4 | — | |
WPZVXHODDBZCLI
|
7.1 | Ki | 4 | — | |
ALKYWGCWYLWWQX
|
6.9 | Ki | 4 | — | |
CHSWXCHUJHYZLB
|
6.9 | Ki | 4 | — | |
ICMPUUKPBRMOSD
|
6.9 | Ki | 4 | — | |
XIHRZTWKTVFWSV
|
6.9 | Ki | 4 | — | |
ANHXASYJLDAVKI
|
6.8 | Ki | 4 | — | |
GREDJTIKEQWSJW
|
6.7 | Ki | 4 | — | |
RYVHKZGUULZSGD
|
6.7 | Ki | 4 | — | |
CLTYJDDMFQEKEL
|
6.0 | Ki | 6 | — | |
QMAXHSLPLMYIPN
|
6.0 | Ki | 6 | — |