Target Details
| UniProt AC | Q16539 |
|---|---|
| Gene Symbol | MAPK14 |
| Protein Name | Mitogen-activated protein kinase 14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,754
- Clinical molecules 97
- Avg pChEMBL 7.28
KEGG Pathways (65)
- AGE-RAGE signaling pathway in diabetic complications
- Adrenergic signaling in cardiomyocytes
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Cellular senescence
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Kaposi sarcoma-associated herpesvirus infection
- Leishmaniasis
- Leukocyte transendothelial migration
- Lipid and atherosclerosis
- MAPK signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Neutrophil extracellular trap formation
- Non-alcoholic fatty liver disease
- Oocyte meiosis
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathogenic Escherichia coli infection
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platelet activation
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Proteoglycans in cancer
- RIG-I-like receptor signaling pathway
- Rap1 signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- Sphingolipid signaling pathway
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Thermogenesis
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- VEGF signaling pathway
- Yersinia infection
Active Molecules (1,754)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FDOKUBCOHMHXDS
|
7.8 | IC50 | 2 | — | |
KWAVLFMTWZNHCQ
|
7.8 | IC50 | 2 | — | |
NVUCXTBAGHPGKH
|
7.8 | IC50 | 2 | — | |
PDRRMIHGJSJJLS
|
7.8 | IC50 | 3 | — | |
ROYXMGVXIACORO
|
7.8 | IC50 | 4 | — | |
SCDOWHQVNDXVPB
|
7.8 | IC50 | 3 | Yes | |
SZGSGJYBCFJTQE
|
7.8 | IC50 | 2 | — | |
VSQDAQJVIALSGZ
|
7.8 | IC50 | 3 | — | |
XBFRRCZSSOFGAI
|
7.8 | IC50 | 3 | — | |
ZMUWOLHXXFLWAH
|
7.8 | IC50 | 2 | — | |
BANXPZGDYGVXOC
|
7.8 | IC50 | 4 | — | |
DGDQMZKPMBIFOF
|
7.8 | IC50 | 4 | — | |
KRAOZXBAPOLPAO
|
7.8 | IC50 | 4 | — | |
LJAUTNHJCPVWDZ
|
7.8 | IC50 | 3 | — | |
NADBSABGTQOEQF
|
7.8 | IC50 | 2 | — | |
OIENACMNANMKKJ
|
7.8 | IC50 | 2 | — | |
OXVQEZJDLGHTQA
|
7.8 | IC50 | 2 | — | |
XIPYKUQAZQIESI
|
7.8 | IC50 | 2 | — | |
NVHXKPSEDLLPHV
|
7.8 | IC50 | 2 | — | |
PDLLDHAITUYAEV
|
7.8 | IC50 | 2 | — | |
AFZIRKJTSPMVSW
|
7.7 | IC50 | 3 | — | |
BMJIPGXVDYVSGD
|
7.7 | IC50 | 4 | — | |
DFRPRNRPOSSJQZ
|
7.7 | IC50 | 2 | Yes | |
HTMINSIGYJFGEU
|
7.7 | IC50 | 3 | — | |
KFJCYTXMHLMPLW
|
7.7 | IC50 | 3 | — | |
OIUJKHYYCHMFEB
|
7.7 | IC50 | 2 | — | |
POOFOKSCEYCHJC
|
7.7 | IC50 | 3 | — | |
SNHWMEWYAPKRQL
|
7.7 | IC50 | 4 | — | |
TUROENOKNBFMBG
|
7.7 | IC50 | 2 | — | |
UNPCCYFJMCHROL
|
7.7 | IC50 | 2 | — | |
VARYUMXVRFFXLR
|
7.7 | IC50 | 3 | — | |
VZONEKWHHXKRRX
|
7.7 | IC50 | 2 | — | |
WSBSGWDWALJLJA
|
7.7 | IC50 | 2 | — | |
BHOZITIWJBGALO
|
7.7 | IC50 | 2 | — | |
BLAZPRXMAUDJQB
|
7.7 | IC50 | 3 | — | |
BLAZPRXMAUDJQB
|
7.7 | IC50 | 3 | — | |
JOIVAEYUULQRLW
|
7.7 | IC50 | 2 | — | |
JVJCVRPAUUWRBH
|
7.7 | Kd | 4 | — | |
NZIUKWCXTXDJLH
|
7.7 | IC50 | 4 | — | |
OTQOZFYTAOFNOL
|
7.7 | IC50 | 3 | — | |
OVYDMAPDQBLTLW
|
7.7 | IC50 | 2 | — | |
PILZXNUZIFIDSU
|
7.7 | IC50 | 3 | — | |
SRMKBWXYOWWDPG
|
7.7 | IC50 | 2 | — | |
VSPFURGQAYMVAN
|
7.7 | IC50 | 17 | — | |
KXQAYIADFSNSAJ
|
7.7 | IC50 | 2 | — | |
DDKMTWFWDUOVDY
|
7.7 | IC50 | 2 | — | |
FIGWQDHDUNOAHY
|
7.7 | IC50 | 2 | — | |
FPWCREKHIZDTGO
|
7.7 | IC50 | 3 | — | |
FSSVIZLKIGCSBI
|
7.7 | IC50 | 3 | — | |
HSODWQGVXRNOEV
|
7.7 | IC50 | 3 | — |