Target Details
| UniProt AC | Q16513 |
|---|---|
| Gene Symbol | PKN2 |
| Protein Name | Serine/threonine-protein kinase N2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02185 (HR1) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 219
- Clinical molecules 15
- Avg pChEMBL 6.87
KEGG Pathways (3)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHGPYYFCIAISBU
|
7.4 | Ki | 31 | — | |
LPILBMJJRGTKOQ
|
7.4 | Ki | 27 | — | |
RJZDECGDCKOHBV
|
7.4 | Ki | 70 | — | |
SKKRZILJUKYLJS
|
7.4 | Ki | 25 | — | |
SLKCVFPEQGHNSI
|
7.4 | Ki | 29 | — | |
VGNKOJURPOHWJF
|
7.4 | Ki | 21 | — | |
ZKHDDJKHTPLPOQ
|
7.4 | Ki | 62 | — | |
MWKSRKSEWLRPBL
|
7.4 | Kd | 1075 | — | |
FQYKIBPUNQVZRF
|
7.4 | IC50 | 2 | — | |
KUVNSIJSYBSMJX
|
7.3 | Ki | 5 | — | |
MLGGUGPIWDHBAI
|
7.3 | IC50 | 10 | — | |
MLGGUGPIWDHBAI
|
7.3 | Ki | 33 | — | |
RFBPWKMQWSIPEO
|
7.3 | Ki | 28 | — | |
SHENEEFOURUIBP
|
7.3 | Ki | 29 | — | |
ZKLJKKASNXVQBZ
|
7.3 | Ki | 27 | — | |
KSKYRXFKNPXFGI
|
7.2 | IC50 | 6 | — | |
DQPYZHUAILXFJI
|
7.2 | Ki | 27 | — | |
LACOMQAWPSFXQC
|
7.2 | Ki | 27 | — | |
QAJPIJHWTGPUNZ
|
7.2 | Ki | 37 | — | |
TVUWQDLBEOZVOU
|
7.2 | Ki | 41 | — | |
VXYDJXMHISGSDA
|
7.2 | Ki | 59 | — | |
HIUHVDROHDSKTC
|
7.1 | Ki | 20 | — | |
IJNGXROUMFEKDB
|
7.1 | Ki | 39 | — | |
JRVSFZKYQCETAH
|
7.1 | Ki | 19 | — | |
LCHCSKHPVCDXAU
|
7.1 | Ki | 30 | — | |
OWRXHGAFWZFFCW
|
7.1 | Ki | 113 | — | |
YPJJSXBVVGPFHA
|
7.1 | Ki | 18 | — | |
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
ACSYKUPGCXYRRO
|
7.0 | Ki | 26 | — | |
AIQDZMUPVYDVLB
|
7.0 | Ki | 48 | — | |
BPNUQXPIQBZCMR
|
7.0 | Ki | 60 | — | |
IYOZTVGMEWJPKR
|
7.0 | Ki | 10 | — | |
JWQOJVOKBAAAAR
|
7.0 | Ki | 29 | — | |
MUKIIGVLQHTSFA
|
7.0 | IC50 | 2 | — | |
RFVBRKXQYUDGIO
|
7.0 | Ki | 23 | — | |
VVEGARMQKNYDID
|
7.0 | Ki | 24 | — | |
SAGGCAPQVJYEGE
|
7.0 | IC50 | 3 | — | |
CNQGNADBGYCKKV
|
6.9 | Ki | 25 | — | |
HOBMVEVXDIOMDM
|
6.9 | Ki | 18 | — | |
MASJMHFQMYAPJR
|
6.9 | Ki | 41 | — | |
MVJMMLFMPWITEJ
|
6.9 | Ki | 110 | — | |
PFCUZXCHLYIMTJ
|
6.9 | Ki | 18 | — | |
ZCXXFPLQFFRMPN
|
6.9 | Ki | 12 | — | |
PBCZSGKMGDDXIJ
|
6.8 | Kd | 68 | Yes | |
VXBAJLGYBMTJCY
|
6.8 | Kd | 34 | Yes | |
ZVSNSFQQKSZZMY
|
6.8 | IC50 | 7 | — | |
DBXGGXLBTWZXBB
|
6.8 | Ki | 39 | — | |
LSLPDHNUWRDOGC
|
6.8 | Ki | 25 | — | |
NGDNKYRUKIPCLK
|
6.8 | Ki | 12 | — | |
SRONQUHCRFZABC
|
6.8 | Ki | 28 | — |