Target Details
| UniProt AC | Q16478 |
|---|---|
| Gene Symbol | GRIK5 |
| Protein Name | Glutamate receptor ionotropic, kainate 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd) |
Summary
- Multi-target molecules 15
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (3)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AXXYLTBQIQBTES
|
9.6 | Ki | 4 | — | |
ZNCDBRBMBIJVRT
|
8.5 | Ki | 4 | — | |
AEKIJKSVXKWGRJ
|
8.0 | Ki | 4 | — | |
PPGDECVBLABBED
|
7.7 | Ki | 4 | — | |
UBGQQPPNOYSQQD
|
7.5 | Ki | 4 | — | |
HEHLSRRDKJVHOM
|
7.2 | Ki | 4 | — | |
ONWXFZVXNOZZFR
|
7.2 | Ki | 9 | — | |
VLSMHEGGTFMBBZ
|
7.1 | Ki | 5 | — | |
PIWNUFICDRESOQ
|
7.0 | Ki | 9 | — | |
YXQUINDTMKETDY
|
7.0 | Ki | 9 | — | |
IEBVITXSHAFLJR
|
6.4 | Ki | 4 | — | |
KTYABWSAGQKAPP
|
6.4 | Ki | 9 | — | |
WYJNVGSFRNBGEH
|
6.2 | Ki | 9 | — | |
WHUUTDBJXJRKMK
|
6.1 | Ki | 5 | — | |
WHUUTDBJXJRKMK
|
6.1 | Ki | 20 | — |