Target Details
| UniProt AC | Q16445 |
|---|---|
| Gene Symbol | GABRA6 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 398
- Clinical molecules 0
- Avg pChEMBL 7.33
KEGG Pathways (8)
Active Molecules (398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HXXGVDKGNHCARX
|
6.6 | IC50 | 16 | — | |
SEWXZWMBVGJJPG
|
6.6 | Ki | 7 | — | |
VMNYVCMDPUOQEL
|
6.6 | Ki | 16 | — | |
GXFWOMYQHNODFA
|
6.6 | IC50 | 16 | — | |
HOTHDLMXYUFPSZ
|
6.6 | IC50 | 16 | — | |
QQONDVXXMVPYIB
|
6.6 | Ki | 16 | — | |
OYXXATFJACEJGE
|
6.6 | Ki | 6 | — | |
GCNSLTKPBZQFJK
|
6.6 | IC50 | 16 | — | |
GQIVRYNNTCEOBX
|
6.6 | Ki | 8 | — | |
ODIZUHKZJZYZAL
|
6.6 | IC50 | 16 | — | |
RTMFRAUTYIKCRK
|
6.6 | Ki | 16 | — | |
QBWJMTOHSYOPBE
|
6.6 | Ki | 7 | — | |
LOFKMRMDVCEZEF
|
6.6 | Ki | 7 | — | |
WNDIDYSCZWXEJF
|
6.6 | Ki | 16 | — | |
LOBNIVNGRUTMOS
|
6.5 | IC50 | 16 | — | |
DLEWDNHPWLPKDJ
|
6.5 | Ki | 8 | — | |
WRUTXEAYYQYJHO
|
6.5 | Ki | 16 | — | |
HJGRBNHROFTASJ
|
6.5 | IC50 | 16 | — | |
KICQPTHJQWBQOI
|
6.5 | Ki | 7 | — | |
QLWLWJVOROKYAO
|
6.5 | Ki | 7 | — | |
YHZXFRGWTKYPKS
|
6.5 | Ki | 16 | — | |
GAQCKHAXURZXGX
|
6.5 | IC50 | 16 | — | |
KNZNHUNBVIKNJP
|
6.5 | Ki | 5 | — | |
HARMZUHRUKGCNG
|
6.5 | Ki | 8 | — | |
VEWLYIAEUXDQBW
|
6.5 | IC50 | 16 | — | |
BCOWBMDVBZPNTD
|
6.5 | Ki | 6 | — | |
GDVGLPNNOCDLLD
|
6.5 | IC50 | 16 | — | |
KDGMRQJYYKGVCJ
|
6.5 | Ki | 7 | — | |
GEFDSAOHFGLQEZ
|
6.5 | Ki | 17 | — | |
UDLTUJYBFNCMJX
|
6.5 | Ki | 7 | — | |
WCTCMHZWHMFZFN
|
6.5 | Ki | 17 | — | |
DDSULWHSYUPHBK
|
6.5 | IC50 | 16 | — | |
XRWYYMUIIXMQBL
|
6.5 | IC50 | 16 | — | |
OOTAQHRUCFIGFZ
|
6.4 | Ki | 7 | — | |
DAYQXLQRTQODQF
|
6.4 | Ki | 16 | — | |
DNCFKDLZZSXXJP
|
6.4 | IC50 | 16 | — | |
MUPIUJYENVWEKT
|
6.4 | IC50 | 16 | — | |
NQFQEBQBZXSXIX
|
6.4 | IC50 | 16 | — | |
VNFZCRPFALLSNM
|
6.4 | IC50 | 16 | — | |
SQPWTARSPNZNEI
|
6.4 | IC50 | 16 | — | |
QCSFXCHHKYXLHE
|
6.4 | Ki | 16 | — | |
YFEZLTPSCJWVHI
|
6.4 | Ki | 16 | — | |
YOJAHANNNITYMX
|
6.4 | Ki | 16 | — | |
ZLAPTIDQRXJQQL
|
6.4 | IC50 | 16 | — | |
AEPFXRGRJZMVIF
|
6.3 | Ki | 17 | — | |
JBTLCAMUYYCXTA
|
6.3 | IC50 | 16 | — | |
DKCNNHVHQYMVTO
|
6.3 | IC50 | 16 | — | |
KKWDMTXJUXKNOU
|
6.3 | Ki | 7 | — | |
BDGWCPYUERFMMY
|
6.3 | Ki | 16 | — | |
UMYWGMKUCZAQJO
|
6.3 | Ki | 16 | — |