Target Details
| UniProt AC | Q16288 |
|---|---|
| Gene Symbol | NTRK3 |
| Protein Name | NT-3 growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13855 (LRR_8) PF16920 (LRRCT_2) PF01462 (LRRNT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 503
- Clinical molecules 19
- Avg pChEMBL 7.52
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (503)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AIWDHNDUIDAYMO
|
6.6 | IC50 | 4 | — | |
ABFNRJFFINRBRG
|
6.5 | IC50 | 2 | — | |
AYXVSCVVQIADBF
|
6.5 | Ki | 10 | — | |
CACMTVGXYAZZNY
|
6.5 | Ki | 11 | — | |
CLRFYTGANQZOBS
|
6.5 | Ki | 41 | — | |
FDVSOQRNTAPCHB
|
6.5 | Ki | 40 | — | |
IZAVTOABECKIDH
|
6.5 | Ki | 20 | — | |
JRLSUZIPUYDUKX
|
6.5 | Ki | 22 | — | |
JSDGKSMNPHJDFK
|
6.5 | Ki | 35 | — | |
NMWSFHOBJVDICZ
|
6.5 | Ki | 2 | — | |
NSYXCWYWACQNOH
|
6.5 | Ki | 10 | — | |
RTYJMUXLFRYRBU
|
6.5 | Ki | 35 | — | |
TXHOCWWJSGCZLC
|
6.5 | Ki | 18 | — | |
VSVWQTDDGQSGHP
|
6.5 | Ki | 51 | — | |
XSRHBCYNCKAFKS
|
6.5 | Ki | 45 | — | |
ZLVOTRRGLSDLPF
|
6.5 | Ki | 36 | — | |
ZVPDNRVYHLRXLX
|
6.5 | Ki | 35 | Yes | |
OVNZXRKXNRIVBK
|
6.5 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.5 | Kd | 65 | — | |
SBGAHKXLTGCPRN
|
6.4 | IC50 | 4 | — | |
QNABDSWBQJKBHK
|
6.4 | IC50 | 45 | — | |
HHSVICUMCOBRPT
|
6.4 | Ki | 33 | — | |
IOBVCHJTLVPPBR
|
6.4 | Ki | 39 | — | |
LVECPYVAIBNSRV
|
6.4 | Ki | 33 | — | |
OUJZYQBEFNDJQN
|
6.4 | Ki | 71 | — | |
ZGDYBJXDIXVTLV
|
6.4 | Ki | 54 | — | |
ZLHFILGSQDJULK
|
6.4 | Ki | 37 | Yes | |
VGNCTJVAUAZQDJ
|
6.4 | IC50 | 3 | — | |
IBUMDLHZUCXAHU
|
6.4 | IC50 | 2 | — | |
CXVBPWYIUWZVJO
|
6.3 | IC50 | 4 | — | |
DEGILXGFBNYPQN
|
6.3 | IC50 | 2 | — | |
DOLVPVSWTLFZMQ
|
6.3 | Ki | 17 | — | |
DSSRVQAIWBZWON
|
6.3 | Ki | 9 | — | |
HZPACYSNLOCDLW
|
6.3 | Ki | 48 | — | |
NLUPJKQOKWBWFC
|
6.3 | Ki | 69 | — | |
OPRQSQDMYPVYOV
|
6.3 | IC50 | 7 | — | |
RAPYFGJGASETOS
|
6.3 | Ki | 11 | — | |
RQUDPSQQOFAWOC
|
6.3 | IC50 | 2 | — | |
UIRCQOKSJDLYBB
|
6.3 | Ki | 50 | — | |
YACXOXQTGJXYNX
|
6.3 | Ki | 11 | — | |
BLYRPGBSIKAIAU
|
6.3 | IC50 | 24 | Yes | |
KQZFHDUZMBMCMO
|
6.3 | IC50 | 3 | — | |
QUOOWHZYYXJNSD
|
6.3 | IC50 | 3 | — | |
CVWXJKQAOSCOAB
|
6.3 | Kd | 35 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
NYYOAOHKRVOFGH
|
6.2 | IC50 | 5 | — | |
HHZIURLSWUIHRB
|
6.2 | Kd | 57 | Yes | |
MLDQJTXFUGDVEO
|
6.2 | Kd | 85 | Yes | |
AQKQATGZIKRZMQ
|
6.2 | Ki | 16 | — | |
GCBJDOWIQHMCMR
|
6.2 | Ki | 84 | — |