Target Details
| UniProt AC | Q16288 |
|---|---|
| Gene Symbol | NTRK3 |
| Protein Name | NT-3 growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13855 (LRR_8) PF16920 (LRRCT_2) PF01462 (LRRNT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 503
- Clinical molecules 19
- Avg pChEMBL 7.52
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (503)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MYQAUKPBNJWPIE
|
6.9 | Kd | 4 | — | |
OYKPWSZSBLRRPL
|
6.9 | IC50 | 11 | — | |
RBMCJUWMZVILNQ
|
6.9 | IC50 | 3 | — | |
ROWJAVCITQHSST
|
6.9 | IC50 | 3 | — | |
UEFCSGDOOJJXTN
|
6.9 | IC50 | 46 | — | |
VXPOXVOQAFEFFO
|
6.9 | IC50 | 3 | — | |
AEYLJTAIDDIOBA
|
6.9 | Ki | 53 | — | |
CJUJLGFTKBBDMG
|
6.9 | Ki | 9 | — | |
IFQICUARAXVEIQ
|
6.9 | Ki | 18 | — | |
KSVGVUZJQAEMMJ
|
6.9 | IC50 | 3 | — | |
IDTRMLOMEBMZLF
|
6.9 | IC50 | 3 | — | |
JGWRKYUXBBNENE
|
6.9 | IC50 | 11 | — | |
FQGDIYVVDKJSNC
|
6.8 | IC50 | 3 | — | |
YWAOBYAAHVVPGD
|
6.8 | IC50 | 3 | — | |
NPVVAEDMCPEANH
|
6.8 | IC50 | 3 | — | |
AQQWWOMMPDCTLW
|
6.8 | Ki | 10 | — | |
CKFSGFBIQDUWKV
|
6.8 | IC50 | 5 | — | |
CLEGDJQQHUTCOW
|
6.8 | Ki | 43 | — | |
DNFPFLPJDNMARR
|
6.8 | IC50 | 3 | — | |
MFMXAWQGPQXDRJ
|
6.8 | Ki | 27 | — | |
UDFDIIVNIYWXDM
|
6.8 | Ki | 74 | — | |
VZUFUBXNQMEQQR
|
6.8 | IC50 | 2 | — | |
XLFNLJYGUOLEJS
|
6.8 | IC50 | 26 | — | |
XPHWIERLJBFPFV
|
6.8 | Ki | 69 | — | |
YEPNVBNYCRGZRX
|
6.8 | Ki | 26 | — | |
YUOWJICKAJQZLS
|
6.8 | Ki | 35 | — | |
MVCOAUNKQVWQHZ
|
6.7 | Kd | 54 | Yes | |
PIQCTGMSNWUMAF
|
6.7 | Kd | 137 | Yes | |
GCIKSSRWRFVXBI
|
6.7 | Kd | 109 | Yes | |
LQVXSNNAFNGRAH
|
6.7 | Kd | 33 | Yes | |
MASJMHFQMYAPJR
|
6.7 | Ki | 41 | — | |
MMMPFWNSQKXKDX
|
6.7 | Ki | 14 | — | |
QXRJBJVCBQSLTA
|
6.7 | Ki | 29 | — | |
RYAVJHIPOWNWDE
|
6.7 | Ki | 38 | — | |
SBFPHSVZEXSHTL
|
6.7 | Ki | 62 | — | |
VBIYDORVDCFKHM
|
6.7 | Ki | 13 | — | |
PQNIGFMNUHDZKX
|
6.7 | IC50 | 4 | — | |
MPVGZUGXCQEXTM
|
6.7 | Kd | 61 | Yes | |
RALKOVHFGYUBAB
|
6.7 | IC50 | 5 | — | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
ZNMQXOQGTZNCCL
|
6.6 | IC50 | 3 | — | |
CXBBWVXSZINRCS
|
6.6 | Ki | 41 | — | |
DNUARRYUJCTBON
|
6.6 | Ki | 2 | — | |
GWMATETWMAQOFL
|
6.6 | Ki | 36 | — | |
JISZKDFLHFISOW
|
6.6 | Ki | 6 | — | |
LRINYHMQZRENCY
|
6.6 | Ki | 29 | — | |
QXKKPVVOOWBLND
|
6.6 | Ki | 8 | — | |
XKFTZKGMDDZMJI
|
6.6 | Ki | 56 | — | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
SZURKEABSBIIMJ
|
6.6 | IC50 | 5 | — |