Target Details
| UniProt AC | Q16236 |
|---|---|
| Gene Symbol | NFE2L2 |
| Protein Name | Nuclear factor erythroid 2-related factor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03131 (bZIP_Maf) |
Summary
- Multi-target molecules 557
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (7)
Associated Diseases (1)
Top Co-occurrence Targets
- KEAP1 557 shared
Active Molecules (557)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDCHEHCCVZBOPQ
|
6.5 | Ki | 2 | — | |
ZIBASFADUCTBIN
|
6.5 | Kd | 2 | — | |
XZGNDSMASLZOKW
|
6.5 | Kd | 2 | — | |
HFYHADGZFKHPEI
|
6.5 | Kd | 2 | — | |
KFMAODZLDUERIC
|
6.5 | IC50 | 2 | — | |
RLQNZMTXCLPEAY
|
6.5 | IC50 | 2 | — | |
WVSQRZIMQWALJT
|
6.5 | IC50 | 2 | — | |
DEMATFZLTHONLJ
|
6.5 | IC50 | 2 | — | |
LETXLDXBLSTFII
|
6.5 | Ki | 2 | — | |
FQVLNJYKCWMFHE
|
6.5 | Kd | 2 | — | |
AGPNUSGKRZZYOM
|
6.5 | IC50 | 2 | — | |
GAFLTUQDNVDCCP
|
6.5 | IC50 | 2 | — | |
PGUQNCOZLHPNFL
|
6.5 | Ki | 2 | — | |
AHHKLAYCXSMRPD
|
6.5 | Ki | 2 | — | |
CHPSOBPPUURRCQ
|
6.5 | Ki | 2 | — | |
FENMHIDJQSBXDN
|
6.5 | Kd | 2 | — | |
ZSEXZJWRCNQRNZ
|
6.5 | IC50 | 2 | — | |
PNBJKHBPNIRWAS
|
6.5 | Kd | 2 | — | |
NTIBHLDTDUOPSN
|
6.4 | IC50 | 2 | — | |
HPTUBKDOPRIRSX
|
6.4 | IC50 | 2 | — | |
ZCGYURKHEKQNGR
|
6.4 | Ki | 2 | — | |
GEYONVKNHOCFKZ
|
6.4 | IC50 | 2 | — | |
HCKKWFYCCAOKMN
|
6.4 | IC50 | 2 | — | |
BRCQFIYBTBPQSU
|
6.4 | Ki | 2 | — | |
UEJISEAYZCHTIJ
|
6.4 | IC50 | 2 | — | |
LGHHKFPHPRCWRF
|
6.4 | IC50 | 2 | — | |
LSMZAJHSVOPJKX
|
6.4 | IC50 | 2 | — | |
DPXLPUCVKPYNBC
|
6.4 | IC50 | 2 | — | |
AMDAELCCBYMSGM
|
6.3 | IC50 | 2 | — | |
LLTUWAURQHDLMT
|
6.3 | IC50 | 2 | — | |
LVGYMFUVDJGNAA
|
6.3 | Kd | 2 | — | |
TXPZGBQJMBXWJO
|
6.3 | Ki | 2 | — | |
XZIIWNBFZABURQ
|
6.3 | Kd | 2 | — | |
DXPBSUNYPNONNA
|
6.3 | IC50 | 2 | — | |
KTGQNHLFJOVZNG
|
6.3 | Kd | 2 | — | |
PMSGXACIVAJWLR
|
6.3 | IC50 | 2 | — | |
VNXRAXRRKSLTKN
|
6.3 | IC50 | 2 | — | |
XTXLNOCEABZQLG
|
6.3 | Ki | 2 | — | |
SGSUJBJLFXJVFX
|
6.3 | Ki | 2 | — | |
AKQXWJHIWSZQPZ
|
6.3 | IC50 | 2 | — | |
BAPMTSPSGNUDMN
|
6.3 | IC50 | 2 | — | |
BBAQYZLFACJTEU
|
6.3 | IC50 | 2 | — | |
BTPDPSLUOKOLFC
|
6.3 | IC50 | 2 | — | |
CAJHFKZCUUGUSQ
|
6.3 | IC50 | 2 | — | |
CCKFFZWASQCQFD
|
6.3 | IC50 | 2 | — | |
CPQNNJBTSHDTLZ
|
6.3 | IC50 | 2 | — | |
CUENPUOZILZXSI
|
6.3 | IC50 | 2 | — | |
CXZPRQFTYURHET
|
6.3 | IC50 | 2 | — | |
DRSUZWSVWLQHEW
|
6.3 | IC50 | 2 | — | |
FGIULSJBSODLAD
|
6.3 | IC50 | 2 | — |