Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ILAGMDVVNQKKBN
|
7.6 | IC50 | 3 | — | |
KCXYXNRPRRXYDO
|
7.6 | IC50 | 5 | — | |
KPLDMYFFSCWABC
|
7.6 | IC50 | 2 | — | |
RSNPTTSTVMVPKM
|
7.6 | IC50 | 3 | — | |
VAISVTUAPAKOSV
|
7.6 | IC50 | 3 | — | |
XXQHACAXRPGDPN
|
7.6 | IC50 | 5 | — | |
FQYQKMRFHCVLGN
|
7.6 | IC50 | 3 | — | |
NPAKNAXWVZRKLD
|
7.6 | IC50 | 3 | — | |
QUOUXYXJTCBLEF
|
7.6 | IC50 | 3 | — | |
DMCMUHXCIDQFES
|
7.6 | IC50 | 3 | — | |
HORZWCBJHIPTFF
|
7.6 | IC50 | 3 | — | |
KBJMHUHSYLAULW
|
7.6 | IC50 | 3 | — | |
OPDSDRNDYJKMNU
|
7.6 | IC50 | 3 | — | |
ULNXAWLQFZMIHX
|
7.6 | IC50 | 7 | — | |
VVLYHQKMEVSGSR
|
7.6 | IC50 | 3 | — | |
VXNSCJKYRXWZBL
|
7.6 | IC50 | 3 | — | |
XMNFQRNWCHJRPC
|
7.6 | IC50 | 3 | — | |
ZSWAHRFSJOAHGN
|
7.6 | IC50 | 3 | — | |
GVZXYFCBILGQCQ
|
7.6 | IC50 | 3 | — | |
XKZOVUPFXXUUBM
|
7.6 | IC50 | 3 | — | |
YADOWFCNQMVLFN
|
7.6 | IC50 | 3 | — | |
ZNUCFGBUOACYBF
|
7.6 | IC50 | 3 | — | |
SKEJWSYZJDVPDG
|
7.6 | IC50 | 3 | — | |
VOOPZQBLDZVBAT
|
7.6 | IC50 | 3 | — | |
DGZUHZNLUIAYRM
|
7.5 | IC50 | 3 | — | |
PTEACBPVIXPKRL
|
7.5 | IC50 | 3 | — | |
YKKKRDOYUHRXGT
|
7.5 | IC50 | 3 | — | |
ZLEVWZJBARHVGV
|
7.5 | IC50 | 3 | — | |
HYUFYHHIABEMLU
|
7.5 | IC50 | 3 | — | |
MCDUVHPSPUQYPE
|
7.5 | IC50 | 3 | — | |
XFUAFESCBCAXHS
|
7.5 | IC50 | 3 | — | |
YNALWGRJSRAASC
|
7.5 | IC50 | 3 | — | |
ZCKREKXDGMDDHF
|
7.5 | IC50 | 3 | — | |
BLRTZJGHISSYGZ
|
7.5 | IC50 | 3 | — | |
GADTVVUDLGZZRJ
|
7.5 | IC50 | 3 | — | |
KRINQRRYPHNQOX
|
7.5 | IC50 | 3 | — | |
MGRZABWUDJKVOB
|
7.5 | IC50 | 3 | — | |
RZHMGYHYURIAFB
|
7.5 | IC50 | 3 | — | |
ZFYVMADJHCXVAS
|
7.5 | IC50 | 3 | — | |
BUSOJUMONRENJH
|
7.5 | IC50 | 3 | — | |
GSPMBCOSONHTOL
|
7.5 | IC50 | 3 | — | |
JDURFLRZRIOZKA
|
7.5 | IC50 | 3 | — | |
QVNFRQNZBTZXRZ
|
7.5 | IC50 | 3 | — | |
YPMMCNYZKNTTQF
|
7.5 | IC50 | 3 | — | |
YQWNSORSVYFCHQ
|
7.5 | IC50 | 3 | — | |
CNFZHWQJHARDDP
|
7.5 | IC50 | 3 | — | |
JJWAMRZWTGVLGV
|
7.5 | IC50 | 3 | — | |
NJDXLHKURDJQHI
|
7.5 | IC50 | 3 | — | |
PWEZXNVUOLJLMU
|
7.5 | IC50 | 3 | — | |
VJSKJBCRWCKMOV
|
7.5 | IC50 | 3 | — |