Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DULCDCQEAIHKPM
|
7.7 | IC50 | 5 | — | |
FZYCWJYPPHUYEK
|
7.7 | IC50 | 5 | — | |
IDUHGUNBWPHVAI
|
7.7 | IC50 | 5 | — | |
KUJUZLBGRRXLMH
|
7.7 | IC50 | 5 | — | |
LVGCTQDARMZPSW
|
7.7 | IC50 | 5 | — | |
OEOBFVJMSOTVQD
|
7.7 | IC50 | 5 | — | |
ONDFGEDYOOIJBZ
|
7.7 | IC50 | 3 | — | |
WHKQTEVRNINIBA
|
7.7 | IC50 | 3 | — | |
XVRVJNZQOATEAP
|
7.7 | IC50 | 5 | — | |
ZBNBGTVUPQTUCA
|
7.7 | IC50 | 3 | — | |
MQNLWRHIHGURGU
|
7.7 | IC50 | 3 | — | |
AKBQMRUQFZTGJP
|
7.7 | IC50 | 4 | — | |
GYACKHYVMFQXGK
|
7.7 | IC50 | 3 | — | |
IFURXQGNBDRQCZ
|
7.7 | IC50 | 3 | — | |
IOKDMBPWICKAAP
|
7.7 | IC50 | 3 | — | |
KJQQIXDWFFOYEG
|
7.7 | IC50 | 3 | — | |
QOYBYCVGYWVUIM
|
7.7 | IC50 | 3 | — | |
QZTPVNUENBWUPE
|
7.7 | IC50 | 3 | — | |
UQJILZDGBXJNJT
|
7.7 | IC50 | 3 | — | |
ZXNDZMFCNRXLTK
|
7.7 | IC50 | 3 | — | |
VZTRXNJTMMFEKF
|
7.7 | IC50 | 3 | — | |
BZSYVCVLCVILPF
|
7.7 | IC50 | 3 | — | |
CTEOMWHGRNOILB
|
7.7 | IC50 | 3 | — | |
HPODOLXTMDHLLC
|
7.7 | IC50 | 2 | — | |
KQZUHEQOOFRWLT
|
7.7 | IC50 | 3 | — | |
RNBZYKQPAMPZJW
|
7.7 | IC50 | 2 | — | |
ZXYWTCVDQLRSRJ
|
7.7 | IC50 | 6 | — | |
DMNYVPRPVYTJBJ
|
7.7 | IC50 | 3 | — | |
LXODDFRAFZGHBG
|
7.7 | IC50 | 4 | — | |
QQZPDOLPTCRTTD
|
7.7 | IC50 | 4 | — | |
YOHCSVVQVICFEW
|
7.7 | IC50 | 3 | — | |
DKVUMSCTMAHGAJ
|
7.6 | IC50 | 3 | — | |
KDYSIBDFRNPOIK
|
7.6 | IC50 | 3 | — | |
LRPCDMLAUKUYGC
|
7.6 | IC50 | 3 | — | |
PSEJQRPWNPCSRG
|
7.6 | IC50 | 3 | — | |
UATGKUUUDPUKBJ
|
7.6 | IC50 | 3 | — | |
YMXIFPGPERBULN
|
7.6 | IC50 | 3 | — | |
YTCYIIQKVJFDTA
|
7.6 | IC50 | 3 | — | |
JNJZSXUCASLSNL
|
7.6 | IC50 | 4 | — | |
VKTSBOIQJNMQAL
|
7.6 | IC50 | 2 | — | |
DPJNKUOXBZSZAI
|
7.6 | IC50 | 4 | — | |
GKZOZSJJEZDVED
|
7.6 | IC50 | 3 | — | |
QWQHIRBPLPABLE
|
7.6 | IC50 | 3 | — | |
RAHSOQYFNLKCMP
|
7.6 | IC50 | 2 | — | |
VFLXVDWCZHLLLM
|
7.6 | IC50 | 4 | — | |
GSOOGSOSZUQKIR
|
7.6 | IC50 | 3 | — | |
LXRKDAIPQPZDBT
|
7.6 | IC50 | 3 | — | |
MOUJXTHVEKPDLC
|
7.6 | IC50 | 3 | — | |
MYEWLWXCQLGFPC
|
7.6 | IC50 | 3 | — | |
DPMPQZDRSNAUCN
|
7.6 | IC50 | 5 | — |