Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIHKWIRREAUTPG
|
7.9 | IC50 | 3 | — | |
WWHYMGYUZYXMOK
|
7.9 | IC50 | 3 | — | |
CFFRRKGGZFEJCN
|
7.9 | IC50 | 3 | — | |
DJPYZFQNPFZTDU
|
7.9 | IC50 | 3 | — | |
GGUAEXUHPRZDCO
|
7.9 | IC50 | 3 | — | |
IIIOCCSATMOANP
|
7.9 | IC50 | 3 | — | |
IOKAODORPXSHDF
|
7.9 | IC50 | 3 | — | |
KNVKGEUUCFUUIB
|
7.9 | IC50 | 3 | — | |
LCKXPIFVVRMPRZ
|
7.9 | IC50 | 3 | — | |
PFWIHYCYPWGTKC
|
7.9 | IC50 | 3 | — | |
FHAZGSWPENWBHD
|
7.9 | IC50 | 3 | — | |
JAFSAJQTBBSUPY
|
7.9 | IC50 | 3 | — | |
LCEAJAZTHFIGTQ
|
7.9 | IC50 | 3 | — | |
JLQBPFPXOAPVDD
|
7.9 | IC50 | 3 | — | |
PFHDWRIVDDIFRP
|
7.9 | IC50 | 2 | — | |
BBEBUGPCQGKOCR
|
7.8 | IC50 | 4 | — | |
DCANOELGDVKTTQ
|
7.8 | IC50 | 3 | — | |
HGZDFOSXMQEHGD
|
7.8 | IC50 | 3 | — | |
ISMVKBKKWVUXRX
|
7.8 | IC50 | 3 | — | |
IZGKHRJIAQLSSB
|
7.8 | IC50 | 3 | — | |
OVBVSKMULHRPLN
|
7.8 | IC50 | 3 | — | |
YRODTWDCXBRTDY
|
7.8 | Ki | 5 | — | |
KARBWWDFFRFWHY
|
7.8 | IC50 | 3 | — | |
KCSVXFVJXLVYFS
|
7.8 | IC50 | 3 | — | |
NOOTVYAYPNGLDI
|
7.8 | IC50 | 3 | — | |
OSZBNUACSVDTOS
|
7.8 | IC50 | 3 | — | |
ACGUFQYGRFKZGD
|
7.8 | IC50 | 3 | — | |
BGXWGWQDFNTTNZ
|
7.8 | IC50 | 3 | — | |
CXLCYFIVMACFAK
|
7.8 | IC50 | 2 | — | |
FDGNPMJCDIJXOQ
|
7.8 | IC50 | 3 | — | |
HALWGZKFCDHYQE
|
7.8 | IC50 | 3 | — | |
IXOMXHCRZBPDTM
|
7.8 | IC50 | 3 | — | |
KOLUAFMFXXTAKO
|
7.8 | IC50 | 3 | — | |
LKDJPLWWFCYONP
|
7.8 | IC50 | 3 | — | |
MWRIGGWWHYYWPL
|
7.8 | IC50 | 4 | — | |
RNUJULGJVKPSBQ
|
7.8 | IC50 | 3 | — | |
WLTNJUUYILGGNP
|
7.8 | IC50 | 3 | — | |
XQFINGFCBFHOPE
|
7.8 | IC50 | 3 | — | |
CHXQYSSALOBPEV
|
7.8 | Kd | 2 | — | |
KNONDVBPBAVBKN
|
7.8 | IC50 | 3 | — | |
FBXFKRLTSXFVRZ
|
7.8 | IC50 | 5 | — | |
FTIMFONTIARMSZ
|
7.8 | IC50 | 3 | — | |
GDDMEOORUYUIJL
|
7.8 | IC50 | 3 | — | |
JCQDRGZRLNNKJK
|
7.8 | IC50 | 5 | — | |
KBQFGSXTQYZJTA
|
7.8 | IC50 | 3 | — | |
LQRSUXVZQNCRKZ
|
7.8 | IC50 | 5 | — | |
QTPQMGNCWCCIHN
|
7.8 | IC50 | 3 | — | |
QYRDDWOUVQBZGU
|
7.8 | IC50 | 3 | — | |
SSDRNUPMYCFXGM
|
7.8 | IC50 | 2 | — | |
VPWRXOUDVYAELQ
|
7.8 | IC50 | 5 | — |