Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FADJTYGNEWCCFM
|
8.0 | IC50 | 6 | — | |
LEFIDTXWZIANAM
|
8.0 | IC50 | 3 | — | |
QTMIDSFRFMBIMS
|
8.0 | IC50 | 3 | — | |
SSUSQQSGMUELGD
|
8.0 | IC50 | 3 | — | |
YFLOKCLJSQKUIO
|
8.0 | IC50 | 6 | — | |
DLOCERYQNWPSFY
|
8.0 | IC50 | 3 | — | |
RKFGJEQBUNXCBP
|
8.0 | IC50 | 3 | — | |
DRICLSBQZNGRNU
|
8.0 | IC50 | 3 | — | |
GODPEQODUHAZTF
|
8.0 | IC50 | 3 | — | |
IOLOBJVPODMXCY
|
8.0 | IC50 | 3 | — | |
KGWISPRJFRVEGL
|
8.0 | IC50 | 3 | — | |
YFKOXEHKCZNWRK
|
8.0 | IC50 | 3 | — | |
CJYTYLFWFWRYEO
|
8.0 | IC50 | 3 | — | |
YJMBAIMXLQUONI
|
8.0 | IC50 | 3 | — | |
YKDXNDLHEXXOTC
|
8.0 | IC50 | 4 | — | |
GHHHISNURKFXLX
|
8.0 | IC50 | 3 | — | |
IHFLNORWUOBGOO
|
8.0 | IC50 | 3 | — | |
MLSCIYIGMFKQRX
|
8.0 | IC50 | 3 | — | |
OMRNALVBPNPCDM
|
8.0 | IC50 | 2 | — | |
QKZXBIXAKYLFRD
|
8.0 | IC50 | 2 | — | |
QNVHIEQAKJZCLP
|
8.0 | IC50 | 3 | — | |
TZLIDJIDCBJDPA
|
8.0 | IC50 | 3 | — | |
VTHPHTNFFMTPAN
|
8.0 | IC50 | 3 | — | |
WLGNJTZQLMKULW
|
8.0 | IC50 | 3 | — | |
CHAFYTDIKJYPEE
|
8.0 | IC50 | 3 | — | |
ORRSIPZEJAGGKP
|
8.0 | IC50 | 3 | — | |
QCDZWDMYQRCVLA
|
8.0 | IC50 | 2 | — | |
SAWHJBBSBAZMKT
|
8.0 | IC50 | 3 | — | |
AWOMROMVFXGIAA
|
7.9 | IC50 | 3 | — | |
AAMTZISHVXYYHH
|
7.9 | IC50 | 4 | — | |
FKBKWMPYFFCAHA
|
7.9 | IC50 | 3 | — | |
HUPIEZUQZQHDAH
|
7.9 | IC50 | 3 | — | |
OJEZJWDIBGFFMT
|
7.9 | IC50 | 3 | — | |
PZMYACQKVABGEK
|
7.9 | IC50 | 3 | — | |
SYBIETZSDORFFL
|
7.9 | IC50 | 2 | — | |
AQMDZAWSEXSOPJ
|
7.9 | IC50 | 3 | — | |
FSWCLCIVYVNCKT
|
7.9 | IC50 | 3 | — | |
GTPFFCKGIGDQSR
|
7.9 | IC50 | 3 | — | |
MGFRBVQSWCIXFN
|
7.9 | IC50 | 3 | — | |
WMZCIJCAOGMXJT
|
7.9 | IC50 | 3 | — | |
XWBFBLGYMZOMCW
|
7.9 | IC50 | 3 | — | |
YPQWPAMAYXWZLK
|
7.9 | IC50 | 3 | — | |
AVQNQRHKXOPEQK
|
7.9 | IC50 | 3 | — | |
FMKWCZINDLWNKL
|
7.9 | IC50 | 3 | — | |
GNJGTNXXYAEHGW
|
7.9 | IC50 | 4 | — | |
JNGULCGOGGIHKC
|
7.9 | IC50 | 4 | — | |
NECGBMLKHWOUJC
|
7.9 | IC50 | 3 | — | |
OPQWDNJKKMJJBB
|
7.9 | IC50 | 5 | — | |
RHLOKPGCUAJRJZ
|
7.9 | IC50 | 3 | — | |
UCYQQCILVOBLSS
|
7.9 | IC50 | 3 | — |