Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YIFZTYMYYDQEER
|
8.1 | IC50 | 4 | — | |
JDHLVLVHORLDII
|
8.1 | IC50 | 2 | — | |
KEILWHBZYZTFCA
|
8.1 | IC50 | 3 | — | |
LWXVRMZBZZZGRX
|
8.1 | IC50 | 3 | — | |
OXICPRAQBJWTNI
|
8.1 | IC50 | 3 | — | |
RDOJDGMXTYOULW
|
8.1 | IC50 | 3 | — | |
AOIKGMYDDAATGY
|
8.1 | IC50 | 4 | — | |
CQQVPXGIZAZXEE
|
8.1 | IC50 | 3 | — | |
HDNPSWXZXMAXCF
|
8.1 | IC50 | 3 | — | |
HGVOGVKCDOMMKJ
|
8.1 | IC50 | 6 | — | |
HYRXVAVQIHXVFZ
|
8.1 | IC50 | 3 | — | |
LUPMMWSBCIYWFQ
|
8.1 | IC50 | 3 | — | |
XQAVUMLVCNDDEB
|
8.1 | IC50 | 3 | — | |
CSOPDAGIMOCYKX
|
8.1 | IC50 | 3 | — | |
HDRWZYVTIMPROL
|
8.1 | IC50 | 3 | — | |
MCLOYHSXGSUSLW
|
8.1 | IC50 | 4 | — | |
SRAFJKJXDXYIOD
|
8.1 | IC50 | 3 | — | |
DRPIQKNZCVRWMV
|
8.1 | IC50 | 3 | — | |
NSQSAUGJQHDYNO
|
8.1 | IC50 | 6 | — | |
PYGKIPLIGFESER
|
8.1 | IC50 | 3 | — | |
QQOBZPFXQOLKKN
|
8.1 | IC50 | 3 | — | |
QWUVUBIJGXCRJG
|
8.1 | IC50 | 3 | — | |
WCLXXEDRKCRHDV
|
8.1 | IC50 | 3 | — | |
BHBLCFLAEZNRFT
|
8.1 | IC50 | 3 | — | |
DBGJHRRBVXYSJK
|
8.1 | IC50 | 4 | — | |
MYAQSXVDXIGHBQ
|
8.1 | IC50 | 3 | — | |
UBEPSDIRLHHNCK
|
8.1 | IC50 | 4 | — | |
YPAYDYPYAASGSV
|
8.1 | IC50 | 3 | — | |
BVWYYZMMLLMIQW
|
8.1 | IC50 | 3 | — | |
IPNXCHNXDBXYIB
|
8.1 | IC50 | 3 | — | |
ODFHOFSFQGNLAQ
|
8.1 | IC50 | 4 | — | |
PSDUHHKPZROJCO
|
8.1 | IC50 | 3 | — | |
GCXUTKWSOMTREF
|
8.1 | IC50 | 3 | — | |
GUCRIBUTILKTSS
|
8.1 | IC50 | 3 | — | |
OWELJWFIXMPMFU
|
8.1 | IC50 | 3 | — | |
BAPZVZCCTXRUOZ
|
8.1 | IC50 | 3 | — | |
GSGYZQJGPTXSRX
|
8.1 | IC50 | 3 | — | |
ORJYWWNQWIUWOE
|
8.1 | IC50 | 3 | — | |
QUCCBUUUAXXXKV
|
8.1 | IC50 | 4 | — | |
RMTWHRRCJFXDNQ
|
8.1 | IC50 | 3 | — | |
FFLHPNPBWYCDDP
|
8.0 | IC50 | 3 | — | |
UYKAUDISVFXYRM
|
8.0 | IC50 | 3 | — | |
ZDSWQEAIASOXHE
|
8.0 | IC50 | 2 | — | |
BCGJBYDNWMTYIL
|
8.0 | IC50 | 3 | — | |
XXIYZBNCALNBRM
|
8.0 | IC50 | 4 | — | |
PTZXAXMZIQNTIK
|
8.0 | IC50 | 3 | — | |
ZRKQYFJHCJLPNU
|
8.0 | IC50 | 3 | — | |
CYKBBRZJDUAZJW
|
8.0 | IC50 | 3 | — | |
YHLPAOMAIKCDDI
|
8.0 | IC50 | 3 | — | |
CHJLMVBYELJCLC
|
8.0 | IC50 | 2 | — |