Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KUSODWXIHYMVMQ
|
8.2 | IC50 | 3 | — | |
BFHYHNDKUBRSSW
|
8.2 | IC50 | 2 | — | |
FCAXPENQAZDWCQ
|
8.2 | IC50 | 3 | — | |
NYWVSLBALKNFJR
|
8.2 | IC50 | 6 | — | |
WOZANJUBZZPSFE
|
8.2 | IC50 | 3 | — | |
ZGCGVCMUJCQTAY
|
8.2 | IC50 | 3 | — | |
ZTOAAMOSOKIAKY
|
8.2 | IC50 | 6 | — | |
HIOYDIJURIUQHD
|
8.2 | IC50 | 3 | — | |
QXOWLBKQZJYDBS
|
8.2 | IC50 | 3 | — | |
VFTBGQMPOGKNNW
|
8.2 | IC50 | 3 | — | |
XLIBABIFOBYHSV
|
8.2 | IC50 | 3 | — | |
ZOMVWEIFWIFJKG
|
8.2 | IC50 | 3 | — | |
FKIMGKSMUHFYPS
|
8.2 | IC50 | 3 | — | |
PEPPYKUBKDTDCC
|
8.2 | IC50 | 3 | — | |
PZMYACQKVABGEK
|
8.2 | IC50 | 3 | — | |
AZVTZJGVTDJFBH
|
8.2 | IC50 | 3 | — | |
BKNAMNWNBQTSBN
|
8.2 | IC50 | 3 | — | |
FJCBMSWDZOFUHF
|
8.2 | IC50 | 4 | — | |
HFGQPOCPRWCSRT
|
8.2 | IC50 | 2 | — | |
UMZWZXQROIKLCJ
|
8.2 | IC50 | 3 | — | |
LOXNXGMKASZRPN
|
8.2 | IC50 | 3 | — | |
QPPMMEVJOAYDNF
|
8.2 | IC50 | 6 | — | |
DHZFRVBZKIOBEV
|
8.2 | IC50 | 3 | — | |
FZGJUUQXBJOLLZ
|
8.2 | IC50 | 3 | — | |
HRDQQHUKUIKFHT
|
8.2 | IC50 | 2 | — | |
IDFJGFFNCRRYID
|
8.2 | IC50 | 3 | — | |
KRWFLWWFUAILDB
|
8.2 | IC50 | 3 | — | |
NOTLWQUGYNQKIM
|
8.2 | IC50 | 3 | — | |
PVDOHGHDNKZICQ
|
8.2 | IC50 | 3 | — | |
VYUUBEDLACJZLJ
|
8.2 | IC50 | 4 | — | |
ABUKMYSLIKFEPI
|
8.2 | IC50 | 3 | — | |
OWAJZJKXTMXEPC
|
8.2 | IC50 | 3 | — | |
WLVXOPOWSHFTFD
|
8.2 | IC50 | 3 | — | |
XAEZNFSFBSOYDY
|
8.2 | IC50 | 3 | — | |
OXHGVTTVUPZVPG
|
8.2 | IC50 | 3 | — | |
RSKOSZLBEDGTFX
|
8.2 | IC50 | 3 | — | |
XTSFOJUTHMPCOC
|
8.2 | IC50 | 3 | — | |
DMWNOBLGMPUHMK
|
8.2 | IC50 | 3 | — | |
FMPAEGNLXRPGNU
|
8.2 | IC50 | 3 | — | |
KFBDQUMEGVZMJM
|
8.2 | IC50 | 3 | — | |
NNXSOVFXQIVDBQ
|
8.2 | IC50 | 3 | — | |
PTTBRTCFZQRRTL
|
8.2 | IC50 | 3 | — | |
UNASHSXBPRWRBJ
|
8.2 | IC50 | 3 | — | |
HDSWNQKFXBYHKU
|
8.1 | IC50 | 3 | — | |
ILOVEZKDAAUEIT
|
8.1 | IC50 | 2 | — | |
KBQYYXDCPRZITN
|
8.1 | IC50 | 2 | — | |
MPGWCMHQERYODZ
|
8.1 | IC50 | 3 | — | |
QCAPCQDNAVGQLT
|
8.1 | IC50 | 3 | — | |
QQNPDWBNYQVGAI
|
8.1 | IC50 | 3 | — | |
VCMDFQHVNRLVEX
|
8.1 | IC50 | 2 | — |