Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RFMNSTSDHNUZJK
|
8.4 | IC50 | 2 | — | |
DNXQPHQAMCRLAS
|
8.4 | IC50 | 3 | — | |
KIRCKTNYAUIENF
|
8.4 | IC50 | 4 | — | |
KNCHKNZBONBSSY
|
8.4 | IC50 | 3 | — | |
AAJAVYJCVGGOEZ
|
8.4 | IC50 | 3 | — | |
NBLSSBXVTJFIFV
|
8.4 | IC50 | 3 | — | |
ZQROGAWPFDGNBR
|
8.4 | IC50 | 3 | — | |
DGNBZQIVGFSZMN
|
8.4 | IC50 | 3 | — | |
DHAGTXOTXDTYPM
|
8.4 | IC50 | 4 | — | |
FUNZVDGKJVAOOJ
|
8.4 | IC50 | 3 | — | |
RRBVSADYEIGTME
|
8.4 | IC50 | 3 | — | |
CVWPNABDQLFDLZ
|
8.4 | IC50 | 2 | — | |
GQWNHQPLIIQMHA
|
8.4 | IC50 | 3 | — | |
GDFWTTPBIQSHHT
|
8.3 | IC50 | 4 | — | |
IFVFSVNBFOUDSB
|
8.3 | IC50 | 3 | — | |
JOAXXJJQMAVHPP
|
8.3 | IC50 | 3 | — | |
OCESHTFWRIZNHJ
|
8.3 | IC50 | 3 | — | |
SWCUAUVZXOKFQG
|
8.3 | IC50 | 3 | — | |
WECHVOOMMFZEJW
|
8.3 | IC50 | 4 | — | |
YJGGHCUWIOSYKC
|
8.3 | IC50 | 3 | — | |
YPYQBBHVZWUEJU
|
8.3 | IC50 | 3 | — | |
AWFUDKRHSVVXNQ
|
8.3 | IC50 | 4 | — | |
CDQFTBVKAAGOCB
|
8.3 | IC50 | 4 | — | |
HMTITUFTVCNPRK
|
8.3 | IC50 | 3 | — | |
CLWFDFUVIUSTHL
|
8.3 | IC50 | 3 | — | |
HCKCPOSCZKRALI
|
8.3 | IC50 | 3 | — | |
PMNFISMZZAVMSE
|
8.3 | IC50 | 4 | — | |
ATHKBEKKKUVVAJ
|
8.3 | IC50 | 3 | — | |
TXRLRLBNYXSZGD
|
8.3 | IC50 | 3 | — | |
DMOUAYZQHPZOBL
|
8.3 | IC50 | 3 | — | |
LXAVJONJUUHXQC
|
8.3 | IC50 | 3 | — | |
SUJIBUUZBLLTLI
|
8.3 | IC50 | 2 | — | |
VLGDZXFHUXKWIS
|
8.3 | IC50 | 3 | — | |
WZZICXXQMQLPFR
|
8.3 | IC50 | 3 | — | |
YYISXYQDJFLQEA
|
8.3 | IC50 | 3 | — | |
CHJLMVBYELJCLC
|
8.3 | IC50 | 2 | — | |
MJSHEKQQEQBILQ
|
8.3 | IC50 | 3 | — | |
CFZVHLDMRCTMQP
|
8.3 | IC50 | 3 | — | |
DBKOXSUBPPSSOQ
|
8.3 | IC50 | 3 | — | |
FROQSIVUBJGRBJ
|
8.3 | IC50 | 3 | — | |
GPOYFENWQYULOI
|
8.3 | IC50 | 3 | — | |
GYXUFRNFFVEZAF
|
8.3 | IC50 | 4 | — | |
KINCYOIHPUNFIT
|
8.3 | IC50 | 3 | — | |
MNNUANXCGONYRO
|
8.3 | IC50 | 3 | — | |
PGHXHERVUQFEHT
|
8.3 | IC50 | 4 | — | |
BFNBFIAGUDLBGV
|
8.3 | IC50 | 3 | — | |
RKAQCAZCQNMZBG
|
8.3 | IC50 | 3 | — | |
RKNILAHTNIOQKB
|
8.3 | IC50 | 4 | — | |
SAXBCTJESUGKOB
|
8.3 | IC50 | 3 | — | |
CZSNMOPTOAOXSM
|
8.2 | IC50 | 4 | — |