Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVPNALZXLPFBHR
|
6.5 | IC50 | 5 | — | |
RELJOVYVSLYYAF
|
6.5 | IC50 | 5 | — | |
RJZWPKDRILLWOY
|
6.5 | IC50 | 5 | — | |
RMUQMIXHRVWFLW
|
6.5 | IC50 | 5 | — | |
RYCSQEVYKFGMDL
|
6.5 | IC50 | 5 | — | |
SGPQSSIOHDGUMV
|
6.5 | IC50 | 5 | — | |
SMHLMPSZVTVQDP
|
6.5 | IC50 | 5 | — | |
SMOGNKYOJRPLBS
|
6.5 | IC50 | 5 | — | |
SSPXUFXDBGMUJX
|
6.5 | IC50 | 5 | — | |
TWYPHVCCCUCUHQ
|
6.5 | IC50 | 5 | — | |
UJORTQXRCVKJIH
|
6.5 | IC50 | 5 | — | |
ULCAYNNEZLTPSJ
|
6.5 | IC50 | 5 | — | |
UNEPUTDIPANHMW
|
6.5 | IC50 | 5 | — | |
UVKFNNHKXWKUBX
|
6.5 | IC50 | 5 | — | |
VPOTVMSZBLPUBY
|
6.5 | IC50 | 5 | — | |
WCMWUOKIGJJBEW
|
6.5 | IC50 | 5 | — | |
WEZXQKRCSWEEJV
|
6.5 | IC50 | 5 | — | |
WFYHTTBNCRIVNL
|
6.5 | IC50 | 5 | — | |
WUFADHRATSOXBZ
|
6.5 | IC50 | 5 | — | |
WVAWYXLXRBQNHE
|
6.5 | IC50 | 5 | — | |
XLQNMGXKIXDYJN
|
6.5 | IC50 | 5 | — | |
YAGRWOSMKWMLKY
|
6.5 | IC50 | 5 | — | |
YEMHYUOUSNCKFN
|
6.5 | IC50 | 5 | — | |
YFVGSCVBPNBEPB
|
6.5 | IC50 | 5 | — | |
YNCFEDAZGLIDEG
|
6.5 | IC50 | 5 | — | |
YPCJINHFCMZDAQ
|
6.5 | IC50 | 5 | — | |
YQGZSHFBWVKMJT
|
6.5 | IC50 | 5 | — | |
YUVQFUKCWVZXOX
|
6.5 | IC50 | 5 | — | |
YWKQPPBXESIUPC
|
6.5 | IC50 | 5 | — | |
YXCILEJYVNSKQL
|
6.5 | IC50 | 5 | — | |
ZDBPLSPFJZAYOW
|
6.5 | IC50 | 5 | — | |
ZDQJJBMRCPYHGA
|
6.5 | IC50 | 5 | — | |
ZIPIJERVXUXJAA
|
6.5 | IC50 | 5 | — | |
ZMBBZQDNQSEFTN
|
6.5 | IC50 | 5 | — | |
ZTFMSQSTAHJAPT
|
6.5 | IC50 | 5 | — | |
ZZGXEORREMDNQW
|
6.5 | IC50 | 5 | — | |
PRHRGMYBHVSWIV
|
6.5 | IC50 | 4 | — | |
COZZQLDZHGRLSF
|
6.5 | IC50 | 4 | — | |
FOOXUZRFPGZBNI
|
6.5 | IC50 | 5 | — | |
LVGCTQDARMZPSW
|
6.5 | IC50 | 5 | — | |
MMBRIKLEHZRKNB
|
6.5 | IC50 | 5 | — | |
QZNVCDCOFCNGGK
|
6.5 | IC50 | 5 | — | |
DSRGQUAKJMFUEU
|
6.5 | IC50 | 4 | — | |
ZJUKTBDSGOFHSH
|
6.5 | IC50 | 22 | — | |
BMOCCPFBSUUTKQ
|
6.5 | IC50 | 4 | — | |
UOZNOEFRBLMVOE
|
6.5 | IC50 | 4 | — | |
WSWAVUBNGPYQHJ
|
6.5 | IC50 | 4 | — | |
IHPVMYOGNXSUKI
|
6.4 | IC50 | 4 | — | |
HCZPNALPIXSQEE
|
6.4 | IC50 | 5 | — | |
SSGKOEJSQSFNGA
|
6.4 | IC50 | 5 | — |