Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTZWAJBMXDSNSI
|
7.1 | IC50 | 3 | — | |
FRTKPKWRJMIGMN
|
7.1 | IC50 | 5 | — | |
OMKHWTRUYNAGFG
|
7.1 | IC50 | 2 | — | |
SPEWFOBJMMAASC
|
7.1 | IC50 | 5 | — | |
NFECTNKYOSHSKZ
|
7.1 | IC50 | 2 | — | |
QHQAGMSQHMYPIY
|
7.1 | IC50 | 3 | — | |
ZAAPADHDHFHGBM
|
7.1 | IC50 | 4 | — | |
AYJXBDHEKFJJEF
|
7.1 | IC50 | 4 | — | |
YFRHDMLBVJDGBP
|
7.1 | IC50 | 3 | — | |
IJWLKFMTKOETBV
|
7.0 | IC50 | 3 | — | |
JNCVEBKTGSGHRB
|
7.0 | IC50 | 4 | — | |
OXWVJBIVVWVCRX
|
7.0 | IC50 | 4 | — | |
QVRCUVHEAFEEBI
|
7.0 | IC50 | 3 | — | |
CZCQPLWFGOLPPQ
|
7.0 | IC50 | 2 | — | |
DXBZHMRTDJUMEJ
|
7.0 | IC50 | 5 | — | |
FNOJLACFKLOHLN
|
7.0 | IC50 | 4 | — | |
GZHOTTJMYDUDKU
|
7.0 | IC50 | 5 | — | |
ZOZZQJIESSTKJX
|
7.0 | IC50 | 5 | — | |
DYIRSNMPIZZNBK
|
7.0 | IC50 | 4 | — | |
UMVGGSVJWIAHAH
|
7.0 | IC50 | 4 | — | |
FYQNDJIEIPRDCS
|
7.0 | IC50 | 3 | — | |
DNSRVUFQXXUPCK
|
7.0 | IC50 | 5 | — | |
LSPMPWXPEAEVGD
|
6.9 | IC50 | 4 | — | |
KYFUPLQMKRWTEP
|
6.9 | IC50 | 3 | — | |
BPVVBXTWDZKTIU
|
6.9 | IC50 | 3 | — | |
UJCVLPBWAQOTMZ
|
6.9 | IC50 | 3 | — | |
WITFAJZVQRHUMQ
|
6.9 | IC50 | 5 | — | |
YOHRBCVKYCQQJA
|
6.9 | IC50 | 5 | — | |
XRTLMSCRDZOHHB
|
6.9 | IC50 | 3 | — | |
PIUDMQZOXJMZKR
|
6.8 | IC50 | 5 | — | |
YTHOTLCZYQVYSA
|
6.8 | IC50 | 2 | — | |
KXKHVGAAZDADOY
|
6.8 | IC50 | 3 | — | |
ZOCJIFRFYZKPCJ
|
6.8 | IC50 | 3 | — | |
TZZZJLSKOPRNFT
|
6.8 | IC50 | 3 | — | |
HFPTVKCVVCVGRX
|
6.8 | IC50 | 5 | — | |
LLXDKFMURVBHJV
|
6.8 | IC50 | 5 | — | |
MRSABGAGWFPBGX
|
6.8 | IC50 | 3 | — | |
WZHRHBHKZPCUTK
|
6.8 | IC50 | 4 | — | |
QLTFOHFSLUPAAG
|
6.8 | IC50 | 2 | — | |
UVKAXCAVTAJIHC
|
6.8 | IC50 | 5 | — | |
ISFOOHZGXXVIFR
|
6.7 | IC50 | 3 | — | |
AHMAQXSPEKRSCD
|
6.7 | IC50 | 5 | — | |
FLKYDMHLGCEZDO
|
6.7 | IC50 | 4 | — | |
IZOARSUTSNEABS
|
6.7 | IC50 | 3 | — | |
LZBICHWHSABGJQ
|
6.7 | IC50 | 5 | — | |
MSDIGPXZCVFNIA
|
6.7 | IC50 | 2 | — | |
VKIJWCDJJOLWKH
|
6.7 | IC50 | 5 | — | |
NUXDGTICHKUALT
|
6.7 | IC50 | 4 | — | |
IRSPKVWRIZJRKO
|
6.7 | IC50 | 3 | — | |
KDYLMJROLWJNNS
|
6.7 | IC50 | 4 | — |