Target Details
| UniProt AC | Q15910 |
|---|---|
| Gene Symbol | EZH2 |
| Protein Name | Histone-lysine N-methyltransferase EZH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 847
- Clinical molecules 0
- Avg pChEMBL 7.4
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BCXFQOXVZKGYFG
|
9.5 | IC50 | 2 | — | |
YUGYQZBNPLWZEK
|
9.5 | IC50 | 2 | — | |
HSPAORFDQDFABD
|
9.4 | IC50 | 2 | — | |
HHSSNFZJCXGEOC
|
9.2 | IC50 | 2 | — | |
GWWPLMJVLCHYQG
|
9.1 | IC50 | 6 | — | |
RERIIBOQUJUPDM
|
9.1 | Kd | 2 | — | |
FKSFKBQGSFSOSM
|
9.0 | IC50 | 2 | — | |
AIFGDRAXMCFCSA
|
8.9 | IC50 | 2 | — | |
SLCLWGGPCPYMMD
|
8.9 | IC50 | 2 | — | |
LPDOHGNBHJLAJC
|
8.9 | Kd | 2 | — | |
YLEIVKBLZYEPPM
|
8.9 | Kd | 2 | — | |
DEIZJPMLDLKNGP
|
8.8 | IC50 | 2 | — | |
DLZBXGWPXWPQBZ
|
8.8 | IC50 | 3 | — | |
IZCXXYQSEKORLW
|
8.8 | Kd | 2 | — | |
YRMUTFZXZBHCGR
|
8.8 | IC50 | 4 | — | |
HFFMKDPDYXSYTK
|
8.7 | IC50 | 3 | — | |
MWCOYDBWBFJQIT
|
8.7 | IC50 | 5 | — | |
BERFMMVJMKSJBI
|
8.7 | IC50 | 2 | — | |
SQRUTRRYZYPVRD
|
8.7 | IC50 | 4 | — | |
FKSFKBQGSFSOSM
|
8.6 | IC50 | 4 | — | |
LORVKFYVSXATKW
|
8.6 | IC50 | 5 | — | |
NXSYWBPZACPLLZ
|
8.6 | IC50 | 2 | — | |
SHEHZRMEIPKJAT
|
8.6 | IC50 | 4 | — | |
QOGRURCTGPYQGF
|
8.6 | IC50 | 5 | — | |
LECDCPFYHWKXQN
|
8.6 | IC50 | 6 | — | |
LONVYJSHGSZBQY
|
8.6 | IC50 | 2 | — | |
USPSIVAZJZHYPK
|
8.6 | IC50 | 2 | — | |
VDWOFKQFWQFVOA
|
8.6 | IC50 | 2 | — | |
CEYRQWJRJOGKRR
|
8.5 | IC50 | 4 | — | |
OGEGKWSUMBNLJE
|
8.5 | IC50 | 6 | — | |
HJWBXJNIZAPAHG
|
8.5 | IC50 | 2 | — | |
IBJQZJITWHHCOE
|
8.5 | IC50 | 6 | — | |
WJGTVLNQOSQGAG
|
8.5 | IC50 | 3 | — | |
ASZHVVIUMMWEHQ
|
8.5 | IC50 | 5 | — | |
SOHBSLPUHGZIPL
|
8.5 | IC50 | 3 | — | |
JFNNNNPSWRAASJ
|
8.5 | IC50 | 4 | — | |
MHZXGNDMFMENQD
|
8.5 | IC50 | 3 | — | |
AOXIOWBVFPMBOP
|
8.5 | IC50 | 2 | — | |
DAAVUJYBTSEGIM
|
8.5 | IC50 | 3 | — | |
ZGXXQCAPJPASHX
|
8.5 | IC50 | 4 | — | |
SMFXHNXJTMDNIG
|
8.5 | IC50 | 4 | — | |
VHEZDOOHAYZQOH
|
8.5 | IC50 | 2 | — | |
RXCVUHMIWHRLDF
|
8.5 | IC50 | 2 | — | |
WHIHSTWOZHKCMY
|
8.5 | IC50 | 4 | — | |
YJHCUUIBUCMIFB
|
8.5 | IC50 | 3 | — | |
SFYRATFDIVLMCE
|
8.4 | IC50 | 3 | — | |
SSDRNUPMYCFXGM
|
8.4 | IC50 | 2 | — | |
SUDKBMFBFAGOBI
|
8.4 | IC50 | 4 | — | |
XAYWQJNGHASKNL
|
8.4 | IC50 | 3 | — | |
DTDNVSQMUWBXOK
|
8.4 | IC50 | 3 | — |