Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VDZFYIRHQIKGSV
|
6.8 | IC50 | 2 | — | |
VTFSQDCQGNSRRY
|
6.8 | IC50 | 2 | — | |
QJYSAPCKCOXUFR
|
6.8 | IC50 | 2 | — | |
JWBFMRPLLUIRBB
|
6.8 | IC50 | 2 | — | |
AMSKTYLOKZVQRX
|
6.7 | IC50 | 3 | — | |
APNKIFBEFRZJNR
|
6.7 | IC50 | 2 | — | |
BSAUUXPPXUVRQO
|
6.7 | IC50 | 2 | — | |
CWRBPYURGIMZCJ
|
6.7 | IC50 | 2 | — | |
CZGJOHTUWRUTMS
|
6.7 | IC50 | 2 | — | |
IRHNPUOYGLVXGO
|
6.7 | IC50 | 2 | — | |
RTMCVMRDJMRVQZ
|
6.7 | IC50 | 2 | — | |
VPPJLAIAVCUEMN
|
6.7 | IC50 | 10 | Yes | |
ZDERPCQJJSCVAI
|
6.7 | IC50 | 2 | — | |
HWYCIQPXYXDOBI
|
6.7 | IC50 | 3 | — | |
KYBPOTYVFWNSGS
|
6.7 | IC50 | 8 | — | |
NDLBOYOWPCRMAR
|
6.7 | IC50 | 2 | — | |
OSVWTSSVVMEISV
|
6.7 | IC50 | 2 | — | |
TZUOZTCIJCIQGB
|
6.7 | IC50 | 3 | — | |
VZULMCMVHNUHKQ
|
6.7 | IC50 | 2 | — | |
ZHYFENVYUKWFHL
|
6.7 | IC50 | 3 | — | |
ZOJAVJOACBCGOH
|
6.7 | IC50 | 3 | — | |
IBMZUIVZLBHAMG
|
6.7 | IC50 | 2 | — | |
UZISDSQSQIPNGM
|
6.7 | IC50 | 2 | — | |
JEEZZJOSUGMGIG
|
6.7 | IC50 | 2 | — | |
LEZRONYAEVJQQI
|
6.7 | IC50 | 2 | — | |
ODNOBAVDQFMWME
|
6.7 | IC50 | 2 | — | |
VULIQUPGKLPKIC
|
6.7 | IC50 | 2 | — | |
AWXDDGVMVDUNGA
|
6.7 | IC50 | 2 | — | |
NJKBBVDDLCQVAF
|
6.7 | IC50 | 2 | — | |
VLXRAZFXSRXIRS
|
6.7 | IC50 | 2 | — | |
UJNYFUQRHSEWMI
|
6.7 | IC50 | 2 | — | |
AEOJAAYXUVZZMW
|
6.7 | IC50 | 2 | — | |
ALYSSPGOUMAGSF
|
6.7 | IC50 | 5 | — | |
BVJWKHFIJISOQD
|
6.7 | IC50 | 2 | — | |
GLRINSLMMNMNDA
|
6.7 | IC50 | 2 | — | |
LBNWDFDPQURJAA
|
6.7 | IC50 | 2 | — | |
YDTDFPARVOEQMG
|
6.7 | IC50 | 2 | — | |
YEDAUVHICLPEIJ
|
6.7 | IC50 | 2 | — | |
JWDYVXBLOYZJLX
|
6.7 | IC50 | 2 | — | |
PDRLXIQAZYHBJG
|
6.7 | IC50 | 2 | — | |
KZBXVOINEPFFDK
|
6.6 | IC50 | 2 | — | |
LXEYTAIEXPOZNY
|
6.6 | IC50 | 2 | — | |
NCFGRWURVNNKRV
|
6.6 | IC50 | 2 | — | |
NHSFBZYDYMUCPM
|
6.6 | IC50 | 2 | — | |
PUIQVUPDIYCXBY
|
6.6 | IC50 | 2 | — | |
ROVOFYSXQNIDPA
|
6.6 | IC50 | 2 | — | |
ZBIVKTYZIJLJTE
|
6.6 | IC50 | 2 | — | |
YFLRARPBRFARON
|
6.6 | IC50 | 2 | — | |
LTPHTGJIOPSZAL
|
6.6 | IC50 | 2 | — | |
VXMXACPWGGRFIF
|
6.6 | IC50 | 2 | — |