Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RFZHHXIXCJHZNR
|
7.0 | IC50 | 2 | — | |
SHUSNHMECJFRFW
|
7.0 | IC50 | 2 | — | |
WTPNXRKKYIAOOU
|
6.9 | IC50 | 2 | — | |
CFWANNDTQNLLHL
|
6.9 | IC50 | 2 | — | |
FOXHBDLHQXLGGN
|
6.9 | IC50 | 2 | — | |
HICKPJYJOOIJSI
|
6.9 | IC50 | 2 | — | |
MUEAMLGBSRPYST
|
6.9 | IC50 | 2 | — | |
NNJOTOMAUDKXKD
|
6.9 | IC50 | 2 | — | |
UEAQPOVLANIUKN
|
6.9 | IC50 | 2 | — | |
WPCMGHHEOJLHRM
|
6.9 | IC50 | 2 | — | |
FSDIGHDJKRVNHH
|
6.9 | IC50 | 2 | — | |
MUUIZCFCJVLOGF
|
6.9 | IC50 | 2 | — | |
QFNICIAXNSXIJO
|
6.9 | IC50 | 2 | — | |
CXCZBWCPIJUCFH
|
6.9 | IC50 | 2 | — | |
BEBRFALPYNNCLU
|
6.9 | IC50 | 2 | — | |
CNJHIRPGEOQTTC
|
6.9 | IC50 | 2 | — | |
KBOLMQHKSVRFIL
|
6.9 | IC50 | 2 | — | |
SSECJOYWYAMJRN
|
6.9 | IC50 | 3 | — | |
FNDAXQFHRLFJSB
|
6.9 | IC50 | 2 | — | |
NUSVQLKNXPBOPF
|
6.9 | IC50 | 2 | — | |
XBAKWGXDYRBWJH
|
6.9 | IC50 | 2 | — | |
ZXMZQSSITMSTKQ
|
6.9 | IC50 | 2 | — | |
KPWHRDZTQCXAAK
|
6.9 | IC50 | 2 | — | |
LGABDIUYXJPBQQ
|
6.9 | IC50 | 2 | — | |
LRBXLVFQDQKSDR
|
6.8 | IC50 | 2 | — | |
OEQKFOZNCUDRFU
|
6.8 | IC50 | 2 | — | |
OPJSVGABDUFTOT
|
6.8 | IC50 | 2 | — | |
PZSZWWKYXIGFLI
|
6.8 | IC50 | 2 | — | |
VGRYEIIRDYDLIT
|
6.8 | IC50 | 2 | — | |
LQBHOJPQVSFKSZ
|
6.8 | IC50 | 2 | — | |
NVLCLKSNVBSVHX
|
6.8 | IC50 | 2 | — | |
WFAAJGGDSHOXSH
|
6.8 | IC50 | 2 | — | |
FCGDQYKNRKWJBF
|
6.8 | IC50 | 2 | — | |
GHOSFOBBUGQTRM
|
6.8 | IC50 | 3 | — | |
LPJFOYUXGSRSAK
|
6.8 | IC50 | 2 | — | |
VRRIYZJUSNMZMP
|
6.8 | IC50 | 2 | — | |
RGTQZYMTUVQERN
|
6.8 | IC50 | 2 | — | |
VPQNAOYBUITQEX
|
6.8 | IC50 | 2 | — | |
DXYBEOOKXLMROC
|
6.8 | IC50 | 2 | — | |
GFFRRUFVZMBJGA
|
6.8 | IC50 | 3 | — | |
GRXUKFHZQDPFAI
|
6.8 | IC50 | 2 | — | |
KGXDTVHRHKTTQK
|
6.8 | IC50 | 2 | — | |
LGAIRKZXPYNIQE
|
6.8 | IC50 | 2 | — | |
PRNTWDYZFJXRDP
|
6.8 | IC50 | 2 | — | |
YVVIILBXFPZWHI
|
6.8 | IC50 | 2 | — | |
FDMPUHDISMOMNB
|
6.8 | IC50 | 2 | — | |
DQVWZYVJOHZANB
|
6.8 | IC50 | 2 | — | |
HZXKYOMFVBZNGK
|
6.8 | IC50 | 2 | — | |
JASALYCADJWQID
|
6.8 | IC50 | 2 | — | |
VDKRGTBLHFOGSC
|
6.8 | IC50 | 2 | — |