Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ISXFEVUJMHDJDV
|
7.2 | IC50 | 2 | — | |
NGDMDSQQEVAVIN
|
7.2 | IC50 | 2 | — | |
OEDXJWJKZWZZTK
|
7.2 | IC50 | 2 | — | |
PKUQWTCYGVRGFE
|
7.2 | IC50 | 2 | — | |
RFLSHFCTAZELPZ
|
7.2 | IC50 | 2 | — | |
WXZNLCQMGILZDR
|
7.2 | IC50 | 2 | — | |
NVPMWUPUWBXETR
|
7.2 | IC50 | 2 | — | |
JHTBXYQIHWCGPI
|
7.1 | IC50 | 2 | — | |
OZAUCXKCFJDDRB
|
7.1 | IC50 | 2 | — | |
RCPKTZHXPBTTTM
|
7.1 | IC50 | 2 | — | |
YYWBVRDWEWYDOV
|
7.1 | IC50 | 2 | — | |
FBZQUICLUFAFPQ
|
7.1 | IC50 | 2 | — | |
CUKXCYUCHNHBBC
|
7.1 | IC50 | 2 | — | |
FKGBDYKCOHLSSI
|
7.1 | IC50 | 2 | — | |
BECROBIDPQYXRW
|
7.1 | IC50 | 2 | — | |
NESLCFXDKPAXII
|
7.1 | IC50 | 2 | — | |
REZDHPKOVBPAMP
|
7.1 | IC50 | 2 | — | |
UMLBPTKZCLVUIO
|
7.1 | IC50 | 2 | — | |
YTHVKXJUOMIOFP
|
7.1 | IC50 | 3 | — | |
BDPIGJCLXMOTDZ
|
7.1 | IC50 | 2 | — | |
HLJJNNPHQAQLII
|
7.1 | IC50 | 2 | — | |
NNYFWIVNWYRZQL
|
7.1 | IC50 | 2 | — | |
TZZDBEDTIJHZJP
|
7.1 | IC50 | 2 | — | |
BBSAEKOKKBAQRH
|
7.1 | IC50 | 2 | — | |
CCIDREHXLARDHU
|
7.1 | IC50 | 2 | — | |
OEPNIHKANHUDFT
|
7.1 | IC50 | 3 | — | |
CXSICEXKLUHLDZ
|
7.1 | IC50 | 3 | — | |
FERUCLMBAKQOAA
|
7.1 | IC50 | 2 | — | |
FSOVHPVLGSQHOZ
|
7.1 | IC50 | 2 | — | |
CCPARYWKMKSOGZ
|
7.0 | IC50 | 2 | — | |
GUMIVJFWYYSBKF
|
7.0 | IC50 | 2 | — | |
MXRDODCDBFHGBL
|
7.0 | IC50 | 2 | — | |
PLCCMQZNQDPYTG
|
7.0 | IC50 | 2 | — | |
SHCCRGIIPVJFHB
|
7.0 | IC50 | 2 | — | |
AKEOVDDAHTWBGN
|
7.0 | IC50 | 3 | — | |
CCBSICWZDFRVAU
|
7.0 | IC50 | 2 | — | |
CEHAIZRVGILZFK
|
7.0 | IC50 | 3 | — | |
KEDUVOFLBUTJTP
|
7.0 | IC50 | 2 | — | |
MLUQPNYVJYPKKO
|
7.0 | IC50 | 2 | — | |
ALQOLRCTDNIXDY
|
7.0 | IC50 | 2 | — | |
WTQGKPCUKPVRSK
|
7.0 | IC50 | 2 | — | |
ZDYIMJLPMWNRHT
|
7.0 | IC50 | 2 | — | |
NFUBWILZNIMKMD
|
7.0 | IC50 | 2 | — | |
RUKSBVHNOBYDMK
|
7.0 | IC50 | 2 | — | |
HBEHFCQVYTUQRI
|
7.0 | IC50 | 2 | — | |
CGIIUPAJBKYEQQ
|
7.0 | IC50 | 2 | — | |
HGMBLKLOKFTAOU
|
7.0 | IC50 | 2 | — | |
QLJAUMYWJMHEIG
|
7.0 | IC50 | 2 | — | |
KNUSTXCZNIGYBZ
|
7.0 | IC50 | 2 | — | |
MHEJDCLHINDVMO
|
7.0 | IC50 | 2 | — |