Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYPMZYYZUJQOOS
|
7.4 | IC50 | 2 | — | |
ZBFHVTYUERGXHJ
|
7.4 | IC50 | 2 | — | |
ZECJEHQTOHGKFP
|
7.4 | IC50 | 2 | — | |
ATRLVPLKGMTSHY
|
7.4 | IC50 | 2 | — | |
IJKKZVFOENDHPB
|
7.4 | IC50 | 2 | — | |
VUCGOPZDZHFBHO
|
7.4 | IC50 | 2 | — | |
RJICYSPMHMARFC
|
7.4 | IC50 | 2 | — | |
RVFFHAQSQFHDKW
|
7.4 | IC50 | 2 | — | |
GNEIAVSENMALRU
|
7.4 | IC50 | 3 | — | |
FECNWUDMIMNVGT
|
7.3 | IC50 | 2 | — | |
IQETYCXHLGJUJR
|
7.3 | IC50 | 3 | — | |
MFMKNWRHVZVDBH
|
7.3 | IC50 | 2 | — | |
NGDMDSQQEVAVIN
|
7.3 | IC50 | 2 | — | |
UZMSDLFEGBEWHD
|
7.3 | IC50 | 2 | — | |
FPPPUMRUUDDRRH
|
7.3 | IC50 | 2 | — | |
NSUPANGHWGJPCM
|
7.3 | IC50 | 2 | — | |
VVSUNZXJDARYBH
|
7.3 | IC50 | 2 | — | |
BENAISSLCJROOE
|
7.3 | IC50 | 2 | — | |
DXOIDXNPYTZMEK
|
7.3 | IC50 | 2 | — | |
IRKLGNYNAXCIJW
|
7.3 | IC50 | 2 | — | |
IXXSLXXUOAYZEZ
|
7.3 | IC50 | 2 | — | |
JZGNUJUVVQHLMQ
|
7.3 | IC50 | 2 | — | |
MIOOLADVEXMJRX
|
7.3 | IC50 | 2 | — | |
USTPUKPHUQZTTM
|
7.3 | IC50 | 2 | — | |
XWNXLYNIWAXGBY
|
7.3 | IC50 | 2 | — | |
YYGZVYTVCWHOFB
|
7.3 | IC50 | 2 | — | |
PPKNTGHPZNLOFG
|
7.3 | IC50 | 2 | — | |
BNAUYEHEMNFFCD
|
7.3 | IC50 | 2 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
CSGMIVCOTWOCPC
|
7.3 | IC50 | 2 | — | |
AVOALNAAWZWOQC
|
7.2 | IC50 | 2 | — | |
DTWJNQKJWMKSFE
|
7.2 | IC50 | 2 | — | |
ZKNUWIKFMSHCTJ
|
7.2 | IC50 | 2 | — | |
IAIPNCLMOFPGLW
|
7.2 | IC50 | 2 | — | |
QLRCVALQRZFUQM
|
7.2 | IC50 | 3 | — | |
MVNGCPNFVZJQQK
|
7.2 | IC50 | 3 | — | |
CVUSIJVOABHLEJ
|
7.2 | IC50 | 3 | — | |
JAUQXVXTUFWMRU
|
7.2 | IC50 | 2 | — | |
NEGWWOJFNIDTET
|
7.2 | IC50 | 2 | — | |
UGOYONMBZFCBPL
|
7.2 | IC50 | 2 | — | |
VYGMELUEYAGXCD
|
7.2 | IC50 | 2 | — | |
NJGHOWOIRIXDKZ
|
7.2 | IC50 | 2 | — | |
NUHUWFKTWWXUTJ
|
7.2 | IC50 | 2 | — | |
RIDSJFHKIZEMRJ
|
7.2 | IC50 | 2 | — | |
FCXMXLXAUSDGLN
|
7.2 | IC50 | 2 | — | |
GVJVTZIRACSJPP
|
7.2 | IC50 | 2 | — | |
NEGUYMSGZYTTPG
|
7.2 | IC50 | 2 | — | |
BGEXEHUFMGIZSJ
|
7.2 | IC50 | 2 | — | |
PPMOJHYERWGAEB
|
7.2 | IC50 | 2 | — | |
BJWJWHANJDRZGO
|
7.2 | IC50 | 3 | — |