Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VUDJTKZNZPHLEX
|
8.2 | IC50 | 2 | — | |
WDDGGSNPHYNGMF
|
8.2 | IC50 | 2 | — | |
ZQXXVCXFDRFOAC
|
8.2 | IC50 | 2 | — | |
XUCXIMYTIQZZHZ
|
8.2 | IC50 | 5 | — | |
QCDLGAPJZJODRJ
|
8.2 | IC50 | 2 | — | |
IMUKSSQOUCDNFP
|
8.2 | IC50 | 2 | — | |
XOKHNIWKPBYBRC
|
8.2 | IC50 | 2 | — | |
FYUHLCNXSLHELL
|
8.2 | IC50 | 2 | — | |
KPHLEZXDKXIWFG
|
8.2 | IC50 | 2 | — | |
ZUPILDXMDFYYGB
|
8.2 | IC50 | 2 | — | |
YOMNBFDPZACIQP
|
8.1 | IC50 | 2 | — | |
GRYVZXPJYFDBIS
|
8.1 | IC50 | 2 | — | |
JKTHEHVHKZOFOB
|
8.1 | IC50 | 2 | — | |
NWFSPMULTCJVGD
|
8.1 | IC50 | 2 | — | |
RQJYQECMAVLMJI
|
8.1 | IC50 | 2 | — | |
USIAWHSRJOGWQW
|
8.1 | IC50 | 2 | — | |
XFWKBJBSEOZBRA
|
8.1 | IC50 | 3 | — | |
MYERANCLHZKYQM
|
8.1 | IC50 | 2 | — | |
WJRHMCNOLMTJKY
|
8.1 | IC50 | 3 | — | |
DSSSTXWTCIBGSG
|
8.1 | IC50 | 2 | — | |
HXQNEKJQBGXFAG
|
8.1 | IC50 | 2 | — | |
GGHBVUAXMMWOPA
|
8.1 | IC50 | 3 | — | |
MRGAEPZPKCBOGL
|
8.1 | IC50 | 2 | — | |
GPPTZPCHCLOBIL
|
8.1 | IC50 | 2 | — | |
LWWVWDWLINDCGR
|
8.1 | IC50 | 2 | — | |
RGKGDWOKTINAMY
|
8.1 | IC50 | 2 | — | |
RHNQUMXARXOPCS
|
8.1 | IC50 | 2 | — | |
GHTDSDKXPCEXRT
|
8.0 | IC50 | 2 | — | |
IPKXOBOEJFTCKO
|
8.0 | IC50 | 2 | — | |
HCTZADLXNTVPRR
|
8.0 | IC50 | 2 | — | |
IFRGFTQIIMWCJG
|
8.0 | IC50 | 2 | — | |
MTQBZRRUVZFECS
|
8.0 | IC50 | 2 | — | |
ODMZUCMOJODESH
|
8.0 | IC50 | 2 | — | |
PUJACRUZSBNORY
|
8.0 | IC50 | 2 | — | |
SWQMDMRTGZSDLJ
|
8.0 | IC50 | 2 | — | |
TVQFYGIEBVVYRN
|
8.0 | IC50 | 4 | — | |
WVXWILBXLFSUOH
|
8.0 | IC50 | 2 | — | |
BHJSCRNVDBKWGW
|
8.0 | IC50 | 2 | — | |
DGULQSWQLJIZCW
|
8.0 | IC50 | 2 | — | |
DQMMXAIHRCDFHS
|
8.0 | IC50 | 3 | — | |
GBHRQRRRPLTXEK
|
8.0 | IC50 | 2 | — | |
YCLDIBUXJUIEOU
|
8.0 | IC50 | 2 | — | |
ZYSCOUXLBXGGIM
|
8.0 | IC50 | 9 | — | |
KFLDDFUYNBKZOT
|
7.9 | IC50 | 2 | — | |
DDDJXDIRHGUPLP
|
7.9 | IC50 | 2 | — | |
NCYAOGNZTIDLCT
|
7.9 | IC50 | 3 | — | |
KSBYUWHBUZLDDL
|
7.9 | IC50 | 2 | — | |
DHSOPLGHCCWMQK
|
7.9 | IC50 | 3 | — | |
MLPXAEWHSAPBSG
|
7.9 | IC50 | 2 | — | |
XLJZYUNHARIFIX
|
7.9 | IC50 | 2 | — |