Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VRUSWBLOISBSSJ
|
8.6 | IC50 | 5 | — | |
AOTZMAHOBVGVQU
|
8.6 | IC50 | 3 | — | |
OFMOIJVBLHFGHB
|
8.6 | IC50 | 2 | — | |
YLPZZUYEMQKXPL
|
8.6 | IC50 | 3 | — | |
CIXVIWMKNATLIZ
|
8.5 | IC50 | 3 | — | |
CVHPNFWHLXBWPR
|
8.5 | IC50 | 2 | — | |
DPIPLAYFRAXNRK
|
8.5 | IC50 | 3 | — | |
FPERPEQIXLOVIK
|
8.5 | IC50 | 5 | — | |
GQIRJGCLEQYBML
|
8.5 | IC50 | 3 | — | |
GQIRJGCLEQYBML
|
8.5 | IC50 | 3 | — | |
IPRFOFLOYPAGPA
|
8.5 | IC50 | 2 | — | |
KQJDXTLVXINOPH
|
8.5 | IC50 | 2 | — | |
NEBUOXBYNAHKFV
|
8.5 | IC50 | 5 | — | |
PIGHRURPFWHXDQ
|
8.5 | IC50 | 2 | — | |
QMIHBNPMTMLUMI
|
8.5 | IC50 | 3 | — | |
UNPJOXGIHJVJQC
|
8.5 | IC50 | 2 | — | |
LRYGMRYJDQOKLI
|
8.5 | IC50 | 2 | — | |
MSLIEPIIAJYDTK
|
8.5 | IC50 | 2 | — | |
SDFWLGIHLRLHLP
|
8.5 | IC50 | 3 | — | |
GFDXIUXAFNREKM
|
8.5 | IC50 | 6 | — | |
KDOYGXBJAYKYQW
|
8.5 | IC50 | 2 | — | |
YTSQUJOXQNTPEU
|
8.4 | IC50 | 2 | — | |
REYUORGZKYONMN
|
8.4 | IC50 | 3 | — | |
DPGOQYYAHWEROP
|
8.4 | IC50 | 5 | — | |
JYYKEMPXQHPLKT
|
8.4 | IC50 | 3 | — | |
LBUJARQQUVGRHC
|
8.4 | IC50 | 2 | — | |
LDZNFFGWKHAEMM
|
8.4 | IC50 | 4 | — | |
LKNQEIFVYZPGTP
|
8.4 | IC50 | 2 | — | |
LXWQXQGRQCXLOL
|
8.4 | IC50 | 2 | — | |
OZPDALRKJRELDR
|
8.4 | IC50 | 2 | — | |
ZRPWGKPPPKBYAL
|
8.4 | IC50 | 2 | — | |
KBNXSZUPQRGYNY
|
8.4 | IC50 | 3 | — | |
UTICZDOENGIDOA
|
8.4 | IC50 | 2 | — | |
PMKRZNNFJGGOGE
|
8.4 | IC50 | 2 | — | |
LIJVHEHWJNGQJH
|
8.3 | IC50 | 2 | — | |
IMNAMBYRWSGKHX
|
8.3 | IC50 | 3 | — | |
ADMLHCZRKYFTCM
|
8.3 | IC50 | 2 | — | |
ZWQHQPKNAATKSU
|
8.3 | IC50 | 2 | — | |
DEYOMPPOEBPYPT
|
8.3 | IC50 | 3 | — | |
DLJHITZLSYMCCA
|
8.3 | IC50 | 2 | — | |
ISAZBDJAFDNKIN
|
8.3 | IC50 | 2 | — | |
LRAAZMNBUIISTO
|
8.3 | IC50 | 2 | — | |
YFPFSPWJNLLSJF
|
8.3 | IC50 | 2 | — | |
MWSVLDOKXAVVNZ
|
8.3 | IC50 | 3 | — | |
PRCIGHMFXRYAIG
|
8.2 | IC50 | 3 | — | |
SXOAHIZWCZOILH
|
8.2 | IC50 | 9 | — | |
LLCJMXUOUAGOJT
|
8.2 | IC50 | 3 | — | |
LXEBABFPSLDVID
|
8.2 | IC50 | 2 | — | |
CFMYXEVWODSLAX
|
8.2 | IC50 | 8 | — | |
IKSUDZQUQOMVKP
|
8.2 | IC50 | 2 | — |