Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PNKCJCUVBPXLEN
|
6.2 | IC50 | 2 | — | |
UHOSYFWASOEKPE
|
6.2 | IC50 | 2 | — | |
GFSUVQOECDPIQJ
|
6.2 | IC50 | 4 | — | |
ZDKAXYKVNSBOHU
|
6.2 | IC50 | 2 | — | |
FDUBXBJERWAVTN
|
6.2 | IC50 | 2 | — | |
LSHATFQUHCHGOI
|
6.2 | IC50 | 2 | — | |
MZOPJCMGXOIERS
|
6.2 | IC50 | 2 | — | |
RPQXVSUAYFXFJA
|
6.2 | IC50 | 8 | — | |
RJZQOYOJWXWNKD
|
6.1 | IC50 | 2 | — | |
AOAGKSSQGPUXSO
|
6.1 | IC50 | 2 | — | |
FFXBKKBNWGBOAE
|
6.1 | IC50 | 2 | — | |
NRKTYVBSUNDFEM
|
6.1 | IC50 | 2 | — | |
QUJPVMQGTDABGN
|
6.1 | IC50 | 2 | — | |
RUZRQWYTSWEZCR
|
6.1 | IC50 | 3 | — | |
SSYPIIPRUWAYCB
|
6.1 | IC50 | 2 | — | |
XYCSIKBESLTOLI
|
6.1 | IC50 | 2 | — | |
REGLDXIVBNZLDY
|
6.1 | IC50 | 2 | — | |
JUSUTAPQEPWMEW
|
6.1 | IC50 | 2 | — | |
JFYPAAXJUZZTLT
|
6.1 | IC50 | 3 | — | |
KJFXVAHPAFFCTE
|
6.1 | IC50 | 2 | — | |
RGEBGRLYAPVJLZ
|
6.1 | IC50 | 2 | — | |
WIWJETIDRRVFQC
|
6.1 | IC50 | 2 | — | |
AYTPMWAPDMTVKH
|
6.0 | IC50 | 2 | — | |
MFAWWJPOJNZHOM
|
6.0 | IC50 | 2 | — | |
VFBZQFVDFIBXGZ
|
6.0 | IC50 | 3 | — | |
BHHALVLOZQTWNJ
|
6.0 | IC50 | 2 | — | |
OKFZWUFFIAFNGA
|
6.0 | IC50 | 2 | — | |
PSKAASYIVOPYMH
|
6.0 | IC50 | 2 | — | |
RTLVFTLHWCSMKT
|
6.0 | IC50 | 2 | — | |
INMXDYHKDXGDPC
|
6.0 | IC50 | 2 | — | |
LXNIGQIGUFGETR
|
6.0 | IC50 | 2 | — | |
PDZFTSNLQQQGTI
|
6.0 | IC50 | 2 | — | |
QKPIYVRCVNBYGR
|
6.0 | IC50 | 2 | — | |
KDRVGEHIJOXPBO
|
6.0 | IC50 | 2 | — | |
VATOXHDFJPTCPW
|
6.0 | IC50 | 2 | — | |
WCRBNOREWVLNLP
|
6.0 | IC50 | 2 | — | |
IIZFMAZANLMCRM
|
6.0 | IC50 | 2 | — | |
YNUAEEJQYHYLMS
|
6.0 | IC50 | 2 | — |