Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DYKADKYVLWMPGZ
|
6.6 | IC50 | 2 | — | |
GKCBAIGFKIBETG
|
6.6 | IC50 | 10 | — | |
XJXFPLHCRFQLST
|
6.6 | IC50 | 3 | — | |
HXLNLMXKKIOHJX
|
6.6 | IC50 | 2 | — | |
KLWKJFRXLGLTIH
|
6.6 | IC50 | 4 | — | |
RXHXBPPRDMVRJS
|
6.6 | IC50 | 2 | — | |
WYPZZPOOMZPAJM
|
6.6 | IC50 | 2 | — | |
CGGSZBTXQJLOGP
|
6.6 | IC50 | 3 | — | |
IDVVCBYQIPGRMK
|
6.6 | IC50 | 2 | — | |
PMMALHFQLZXMOO
|
6.6 | IC50 | 2 | — | |
QLKAFHZJICDACE
|
6.6 | IC50 | 3 | — | |
XPZJAEZVONHCRC
|
6.6 | IC50 | 2 | — | |
YUQSIOIGTXTCOF
|
6.6 | IC50 | 3 | — | |
PFHPPXLJMQLSRQ
|
6.6 | IC50 | 2 | — | |
PSTCCBODERRWFK
|
6.6 | IC50 | 2 | — | |
QDYXAAARUBEFCA
|
6.6 | IC50 | 2 | — | |
QKQXMYZOQMBBRN
|
6.6 | IC50 | 2 | — | |
PXKQOZLVZUDGPQ
|
6.5 | IC50 | 2 | — | |
JHSOBKSPKNURCU
|
6.5 | IC50 | 3 | — | |
JUJBEYGCDLLKKZ
|
6.5 | IC50 | 2 | — | |
KHYNGGVKOMNOKG
|
6.5 | Ki | 2 | — | |
ZUXRUQOEFBOTGF
|
6.5 | IC50 | 4 | — | |
ANGUVPSJNSWBFO
|
6.5 | IC50 | 4 | — | |
JFTTWRHSUYMBCX
|
6.5 | IC50 | 2 | — | |
JSPXITPXMRLRIW
|
6.5 | IC50 | 2 | — | |
NSBIALIUYQEBEH
|
6.5 | IC50 | 3 | — | |
OTBNOCRUGHNICR
|
6.5 | IC50 | 2 | — | |
YJMKIYSRJWQPPZ
|
6.5 | IC50 | 2 | — | |
IJZZXHRLQVUZPN
|
6.5 | IC50 | 2 | — | |
JKJROAPYAHIAJY
|
6.5 | IC50 | 2 | — | |
MJJULZATLMLYAP
|
6.5 | IC50 | 2 | — | |
ARJLZIQJKVTPEU
|
6.5 | IC50 | 3 | — | |
KQHRBDBWQHZROV
|
6.5 | IC50 | 3 | — | |
LNYJTKCHVILHMC
|
6.5 | IC50 | 2 | — | |
PJWLKPFEAXQJNQ
|
6.5 | IC50 | 2 | — | |
FIXIITTZIGLTCR
|
6.5 | IC50 | 3 | — | |
WOOZKYJTHJWUFV
|
6.5 | IC50 | 2 | — | |
BBOCRFBJZWHFGM
|
6.5 | IC50 | 2 | — | |
BBOBNSBBLDOMGF
|
6.5 | IC50 | 2 | — | |
NXOLRSKOGVZGJE
|
6.5 | IC50 | 2 | — | |
QWVHTZXEQKODDC
|
6.5 | IC50 | 2 | — | |
JEQHYRZPVUELSI
|
6.4 | IC50 | 2 | — | |
KPACYEJRAQEPQE
|
6.4 | IC50 | 2 | — | |
MHUUDVZSPFRUSK
|
6.4 | Ki | 2 | — | |
MHUUDVZSPFRUSK
|
6.4 | Ki | 2 | — | |
RAXSCIQUOWLHGV
|
6.4 | IC50 | 2 | — | |
RUCRJESLFWTKNO
|
6.4 | IC50 | 2 | — | |
AKAQZLFYNGRABJ
|
6.4 | IC50 | 2 | — | |
RGTQZYMTUVQERN
|
6.4 | IC50 | 2 | — | |
DQVWZYVJOHZANB
|
6.4 | IC50 | 2 | — |