Target Details
| UniProt AC | Q15858 |
|---|---|
| Gene Symbol | SCN9A |
| Protein Name | Sodium channel protein type 9 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 588
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (588)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSPHMGORSRQULF
|
10.8 | IC50 | 6 | — | |
LLEKPWJKKKVEPI
|
9.7 | IC50 | 2 | — | |
OCNOGKDYKRVBCZ
|
9.7 | IC50 | 3 | — | |
PTMJZFRCKPOPSW
|
9.7 | IC50 | 2 | — | |
WWSWLMWIXLNWHP
|
9.7 | IC50 | 2 | — | |
VEEQSZWXUOUXPZ
|
9.6 | IC50 | 5 | — | |
AHWSGUQUIABDFY
|
9.5 | IC50 | 2 | — | |
FQHDBBOTIYOYLF
|
9.5 | IC50 | 3 | — | |
NLTQZTZBFNPMDH
|
9.5 | IC50 | 3 | — | |
DKYUUKRMMHLYCZ
|
9.4 | IC50 | 2 | — | |
MIIOBHGQUATGFU
|
9.4 | IC50 | 2 | — | |
PTCBNPULJWGSML
|
9.4 | IC50 | 9 | — | |
CYBITNCPJFQMIJ
|
9.3 | IC50 | 5 | — | |
AAUMZZJEGXJINE
|
9.3 | IC50 | 3 | — | |
LZJKVSDOJZQQKC
|
9.3 | IC50 | 2 | — | |
NIUMYXYWSPDBFW
|
9.3 | IC50 | 2 | — | |
QEITUNTXHQTCMZ
|
9.3 | IC50 | 2 | — | |
TZPJMFCRZHDJLH
|
9.3 | IC50 | 2 | — | |
XOAUGYVLRSCGBG
|
9.3 | IC50 | 8 | — | |
XQUOWYVEKSXNET
|
9.3 | Kd | 3 | — | |
DFFVMIVCNSUZRH
|
9.2 | IC50 | 2 | — | |
IVVQUXZDEFTOMS
|
9.2 | IC50 | 2 | — | |
SUDPJHWRLKPICV
|
9.1 | IC50 | 3 | — | |
ALEKFWIWCIMWKG
|
9.1 | IC50 | 3 | — | |
KRNHAUPCKRIYSK
|
9.1 | IC50 | 3 | — | |
BQVSSPNOFJNEHA
|
9.0 | IC50 | 2 | — | |
OCGIYHGXHMLCPX
|
9.0 | IC50 | 4 | — | |
KIIZVCWLLOZRPV
|
8.9 | IC50 | 2 | — | |
QGQKYSJJEUMYCP
|
8.9 | IC50 | 2 | — | |
YFFAMHITDBOYET
|
8.9 | IC50 | 2 | — | |
VENWKQHIOIEAII
|
8.8 | IC50 | 3 | — | |
PEIYHGIZJQATLS
|
8.8 | IC50 | 2 | — | |
WGQMMWFPSAVNAJ
|
8.8 | IC50 | 2 | — | |
FCGCWVRBOOKMTK
|
8.7 | IC50 | 3 | — | |
FCGCWVRBOOKMTK
|
8.7 | IC50 | 2 | — | |
GNHZBRMVSAIOCC
|
8.7 | IC50 | 2 | — | |
IFOFQYZJHRNQLW
|
8.7 | IC50 | 2 | — | |
KGGOSMYISLXZHL
|
8.7 | IC50 | 2 | — | |
NBZBSEDIUYZBSR
|
8.7 | IC50 | 2 | — | |
FCTMRPTVPHVTTN
|
8.7 | IC50 | 3 | — | |
GAUCTMQMNSDYNT
|
8.7 | IC50 | 2 | — | |
WQSUNLAAABNZKE
|
8.7 | IC50 | 3 | — | |
KQWOBWMNPNSGDQ
|
8.6 | IC50 | 2 | — | |
XYPYULMUTWWOKW
|
8.6 | IC50 | 2 | — | |
SDFWLGIHLRLHLP
|
8.6 | IC50 | 3 | — | |
YEYOIWDLFZJGMH
|
8.6 | IC50 | 2 | — | |
HRRHRSSCWYTCBS
|
8.6 | IC50 | 3 | — | |
NNBQSDGKUCGYMG
|
8.6 | IC50 | 2 | — | |
AADZPNRBAZVGNN
|
8.6 | IC50 | 2 | — | |
QESPTBXFDDSHIF
|
8.6 | IC50 | 5 | — |