Target Details
| UniProt AC | Q15842 |
|---|---|
| Gene Symbol | KCNJ8 |
| Protein Name | ATP-sensitive inward rectifier potassium channel 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01007 (IRK) PF17655 (IRK_C) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.45
KEGG Pathways (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LVEDGSIMCSQNNX
|
7.1 | IC50 | 4 | — | |
TVZCRIROJQEVOT
|
7.0 | IC50 | 4 | — | |
CBVDKJDKOREVOE
|
6.9 | IC50 | 4 | — | |
PXUHSBKGJFYMON
|
6.4 | IC50 | 4 | — | |
LJLXQHHFAKVTNP
|
6.3 | IC50 | 4 | — | |
LTKRZCMBXQFJLK
|
6.3 | IC50 | 4 | — | |
TVZCRIROJQEVOT
|
6.3 | IC50 | 4 | — | |
GNVWYNKNTYVESS
|
6.3 | IC50 | 4 | — | |
XKQUHPOBIFXEAQ
|
6.2 | IC50 | 4 | — | |
DYMOQRBZQBQYDN
|
6.1 | IC50 | 4 | — | |
XIPHANJESHAHDZ
|
6.1 | IC50 | 4 | — |