Target Details
| UniProt AC | Q15835 |
|---|---|
| Gene Symbol | GRK1 |
| Protein Name | Rhodopsin kinase GRK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 25
- Clinical molecules 10
- Avg pChEMBL 6.51
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
ACLLLJSNOCYQOJ
|
7.3 | IC50 | 8 | — | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
UGYAZGXSMRGKRD
|
7.1 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 147 | Yes | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
NXSJMRCTGYTSTK
|
6.9 | Kd | 200 | — | |
OBZJZDHRXBKKTJ
|
6.7 | Ki | 2 | — | |
GYMOXCZIQHPXOH
|
6.7 | IC50 | 6 | — | |
DMNINFHJFPFPIZ
|
6.6 | IC50 | 4 | — | |
WINHZLLDWRZWRT
|
6.5 | Kd | 201 | Yes | |
XYUFCXJZFZPEJD
|
6.5 | IC50 | 23 | Yes | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
PTJBMQVUHYZJLN
|
6.3 | IC50 | 5 | — | |
KGPGFQWBCSZGEL
|
6.2 | Kd | 59 | Yes | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 82 | Yes | |
HFNKQEVNSGCOJV
|
6.1 | Kd | 65 | — | |
ZCBUQCWBWNUWSU
|
6.1 | Kd | 59 | — | |
HZTYDQRUAWIZRE
|
6.1 | Kd | 40 | Yes | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
XZXHXSATPCNXJR
|
6.0 | Kd | 165 | Yes |